SCHEMBL11633686

SCHEMBL11633686

N#Cc1nc(Cl)c(Sc2ccccc2)nc1C#N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.44
ALDH1A1 P00352 6/20 0.44
CYP1A2 P05177 5/20 0.44
CYP2C9 P11712 5/20 0.44
CYP2C19 P33261 5/20 0.44
MAOA P21397 2/20 0.44
MAOB P27338 2/20 0.44
L3MBTL1 Q9Y468 5/20 0.43
TDP1 Q9NUW8 2/20 0.43
CYP3A4 P08684 3/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HPGD P15428 3/20 0.41
GAA P10253 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 5/20 0.40
ABCG2 Q9UNQ0 1/20 0.37
HTT P42858 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20261932 0.89 MAOA (0.50) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL11004372 0.87 KDM4E (0.47) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL11631447 0.83 CYP1A2 (0.47) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL11630969 0.81 L3MBTL1 (0.52) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL11634112 0.78 ABCG2 (0.46) KDM4EALDH1A1MEN1KMT2ANPSR1
SCHEMBL6376517 0.77 ALDH1A1 (0.50) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL11631356 0.77 AR (0.49) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL11090360 0.75 ALDH1A1 (0.51) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL11095067 0.74 HPGD (0.54) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL9615083 0.74 KDM4E (0.44) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4113724-A Arylthiodicyanopyrazines as plant disease control agents E. I. DU PONT DE NEMOURS AND COMPANY (US) 1978-09-12 US claimed
US-4113724-A Arylthiodicyanopyrazines as plant disease control agents E. I. DU PONT DE NEMOURS AND COMPANY (US) 1978-09-12 US disclosed