SCHEMBL11709161

SCHEMBL11709161

CCOC(=O)C1=C(C)NC(N)=C(C(=O)OCC)C1c1cc(OC)c(OC)c(OC)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.54
KDM4E B2RXH2 2/20 0.54
ALDH1A1 P00352 2/20 0.54
LMNA P02545 1/20 0.54
HPGD P15428 1/20 0.54
HSD17B10 Q99714 1/20 0.54
ADORA3 P0DMS8 3/20 0.50
TSHR P16473 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
ABCC1 P33527 1/20 0.49
CACNA1F O60840 2/20 0.48
CACNA1D Q01668 2/20 0.48
CACNA1S Q13698 2/20 0.48
CACNA1C Q13936 2/20 0.48
UBE2N P61088 1/20 0.46
SIRT3 Q9NTG7 1/20 0.46
SIRT5 Q9NXA8 1/20 0.46
ATM Q13315 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11801987 0.88 GAA (0.54) GAAKDM4EALDH1A1LMNAHPGD
SCHEMBL10849135 0.79 ACHE (0.54) GAAKDM4EALDH1A1LMNAHPGD
SCHEMBL11778065 0.79 UBE2N (0.47) GAAKDM4EALDH1A1LMNAHPGD
SCHEMBL11804240 0.79 SIRT3 (0.50) GAAKDM4EALDH1A1LMNAHPGD
SCHEMBL11522796 0.78 CACNA1D (0.64) GAAKDM4EALDH1A1LMNAHPGD
SCHEMBL10684386 0.78 ADORA3 (0.75) GAAKDM4EALDH1A1LMNAHPGD
SCHEMBL11688373 0.78 DHFR (0.61) GAAKDM4EALDH1A1LMNAHPGD
SCHEMBL14616736 0.76 ADORA3 (0.85) GAAKDM4EALDH1A1LMNAHPGD
SCHEMBL14576820 0.76 ADORA3 (0.68) GAAKDM4EALDH1A1LMNAHPGD
SCHEMBL3028393 0.76 GAA (0.66) GAAKDM4EALDH1A1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4002762-A 2-Amino-3,4-dihydropyridines used to effect coronary vessel dilation and treat hypertension BAYER AKTIENGESELLSCHAFT (DT) 1977-01-11 US disclosed
US-4001252-A HYPOTENSIVES, CORONARY DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1977-01-04 US disclosed