SCHEMBL11713752

SCHEMBL11713752

O=CN1CCN=C(c2ccccc2F)c2cc(Cl)ccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 3/20 0.50
CYP3A4 P08684 3/20 0.50
DRD3 P35462 2/20 0.50
PDE4D Q08499 2/20 0.50
SLC22A1 O15245 1/20 0.50
ABCB11 O95342 1/20 0.50
HTR1A P08908 1/20 0.48
HTR3A P46098 1/20 0.48
KCNH2 Q12809 1/20 0.48
GHSR Q92847 1/20 0.48
LMNA P02545 1/20 0.47
NR1I2 O75469 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
HTR2C P28335 1/20 0.47
ADRA1A P35348 1/20 0.47
PTGS2 P35354 1/20 0.47
CHRNA4 P43681 1/20 0.47
SLC6A3 Q01959 1/20 0.47
CHRM1 P11229 1/20 0.45
SMARCA2 P51531 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11715519 0.89 GABRA1 (0.50) OPRK1PDE4DLMNANR1I2ADORA3
SCHEMBL11716883 0.84 OPRK1 (0.67) OPRK1PDE4DKCNH2LMNANR1I2
SCHEMBL11536241 0.81 OPRK1 (0.70) OPRK1CYP3A4DRD3PDE4DSLC22A1
Hydrochloric Acid SCHEMBL11683071 0.81 OPRK1 (0.69) OPRK1CYP3A4DRD3PDE4DSLC22A1
SCHEMBL11715927 0.80 OPRK1 (0.52) OPRK1CYP3A4DRD3PDE4DSLC22A1
Fletazepam SCHEMBL119540 0.77 CYP3A4 (0.48) OPRK1CYP3A4DRD3PDE4DSLC22A1
SCHEMBL11681501 0.76 CYP3A4 (0.48) OPRK1CYP3A4DRD3PDE4DSLC22A1
SCHEMBL11460301 0.75 SMARCA2 (0.49) OPRK1CYP3A4DRD3PDE4DSLC22A1
SCHEMBL11617590 0.73 CYP3A4 (0.50) OPRK1CYP3A4DRD3PDE4DSLC22A1
SCHEMBL11470290 0.73 CYP3A4 (0.46) OPRK1CYP3A4DRD3PDE4DSLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4002611-A Preparation of benzodiazepines SUMITOMO CHEMICAL COMPANY, LIMITED (JA) 1977-01-11 US disclosed