SCHEMBL11723632

SCHEMBL11723632

Cc1cc(C(F)(F)C(F)(F)F)c2ccc(=O)[nH]c2n1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
ADORA1 P30542 6/20 0.38
ADORA2A P29274 5/20 0.38
PDE2A O00408 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11723044 0.88 AR (0.44) KDM4EKMT2AMEN1ALDH1A1ADORA1
SCHEMBL11716661 0.84 ALDH1A1 (0.35) KMT2AMEN1ALDH1A1PDE2AHTT
SCHEMBL11801511 0.77 KMT2A (0.38) KDM4EKMT2AMEN1ADORA1ADORA2A
SCHEMBL30681004 0.77 ADORA1 (0.47) KDM4EKMT2AALDH1A1ADORA1ADORA2A
SCHEMBL11726649 0.77 KDM4E (0.39) KDM4EKMT2AMEN1ALDH1A1ADORA1
SCHEMBL3320128 0.76 KDM4E (0.64) KDM4EKMT2AMEN1ALDH1A1ADORA1
SCHEMBL11721081 0.71 ALDH1A1 (0.50) KDM4EKMT2AMEN1ALDH1A1HTT
SCHEMBL11724059 0.70 FABP4 (0.43) KDM4EKMT2AMEN1ALDH1A1ADORA1
SCHEMBL13622759 0.67 KDM4E (0.57) KDM4EKMT2AADORA1ADORA2A
SCHEMBL11718448 0.67 KDM4E (0.53) KDM4EKMT2AALDH1A1ADORA1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4031103-A BRONCHODILATOR AGENTS, 2,6-DIAMINOPYRIDINE, DIKETONE COMPOUND MERCK SHARP & DOHME (I.A.) CORPORATION (US) 1977-06-21 US disclosed
US-3962262-A HYPOTENSIVE AGENTS, BRONCHODILATORS MERCK & CO., INC. (US) 1976-06-08 US disclosed