Bromide

Bromide

SCHEMBL1173547

Br.CCN(CC)CCOc1ccccc1

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 known ✓ Q99720 3/20 0.60
CHRM2 known ✓ P08172 2/20 0.60
ADRA2A known ✓ P08913 2/20 0.60
SLC6A2 known ✓ P23975 2/20 0.60
SLC6A4 known ✓ P31645 2/20 0.60
SLC6A3 known ✓ Q01959 2/20 0.60
ADRB3 known ✓ P13945 1/20 0.60
ADRA2B known ✓ P18089 1/20 0.60
ADRA2C known ✓ P18825 1/20 0.60
CHRM3 known ✓ P20309 1/20 0.60
HTR1A known ✓ P08908 1/20 0.60
ADRA1A known ✓ P35348 1/20 0.60
ACHE known ✓ P22303 1/20 0.55
CYP2D6 P10635 2/20 0.72
HTT P42858 2/20 0.72
LTA4H P09960 2/20 0.72
CYP1A2 P05177 1/20 0.72
CYP2C9 P11712 1/20 0.72
CYP2C19 P33261 1/20 0.72
EBP Q15125 3/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1405290 0.98 CYP2D6 (0.74) CYP2D6HTTLTA4HCYP1A2CYP2C9
SCHEMBL12610941 0.98 CYP2D6 (0.74) CYP2D6HTTLTA4HCYP1A2CYP2C9
Hydrochloric Acid SCHEMBL10505479 0.96 CYP2D6 (0.72) CYP2D6HTTLTA4HCYP1A2CYP2C9
SCHEMBL6676718 0.88 LTA4H (0.62) CYP2D6HTTLTA4HCYP1A2CYP2C9
SCHEMBL9706125 0.87 EBP (0.72) CYP2D6HTTLTA4HCYP1A2CYP2C9
SCHEMBL21195812 0.85 KCNA3 (0.64) CYP2D6HTTLTA4HCYP1A2CYP2C9
SCHEMBL22224170 0.85 ALDH1A1 (0.63) CYP2D6HTTLTA4HCYP1A2CYP2C9
Methylamine SCHEMBL10666826 0.85 LTA4H (0.58) CYP2D6HTTLTA4HCYP1A2CYP2C9
SCHEMBL14463907 0.84 LTA4H (0.57) CYP2D6HTTLTA4HCYP1A2CYP2C9
SCHEMBL9706141 0.84 KDM4E (0.73) CYP2D6HTTLTA4HCYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8258328-B2 Method and intermediates for preparing 19-norsteroid compounds AVENTIS PHARMA S.A. (FR) 2012-09-04 US disclosed
US-20110046402-A1 NOVEL METHOD AND INTERMEDIATES FOR PREPARING 19-NORSTEROID COMPOUNDS AVENTIS PHARMA S.A. (FR) 2011-02-24 US disclosed
US-20040229853-A1 Novel method and intermediates for preparing 19-norsteroid compounds AVENTIS PHARMA S.A. (FR) 2004-11-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040229853-A1 Novel method and intermediates for preparing 19-norsteroid compounds CYP17A1, HSD17B7, CYP11B1 SIGMAR1 1097/4885CHRM2 3034/4885ADRA2A 571/4885
US-20110046402-A1 NOVEL METHOD AND INTERMEDIATES FOR PREPARING 19-NORSTEROID COMPOUNDS HSD17B7, CYP17A1, HSD17B13 SIGMAR1 1037/4885CHRM2 1624/4885ADRA2A 412/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.