SCHEMBL11748633

SCHEMBL11748633

CC(=O)c1cc2ccc(OCC(O)CNC(C)(C)C)cc2o1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.53
MEN1 O00255 1/20 0.51
HTT P42858 1/20 0.51
KMT2A Q03164 1/20 0.51
ADRB1 P08588 4/20 0.51
CYP2D6 P10635 2/20 0.50
CASR P41180 3/20 0.48
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA9 Q16790 1/20 0.46
KCNH2 Q12809 2/20 0.46
SLC6A2 P23975 1/20 0.46
SLC6A4 P31645 1/20 0.46
SLC6A3 Q01959 1/20 0.46
ADRB2 P07550 3/20 0.45
EPHX2 P34913 1/20 0.44
ADRB3 P13945 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10512127 0.82 ADRB1 (0.45) CA2MEN1KMT2AADRB1CYP2D6
SCHEMBL11749742 0.77 LMNA (0.54) MEN1KMT2AADRB1CYP2D6KCNH2
SCHEMBL10970320 0.77 ADRB2 (0.53) ADRB1KCNH2ADRB2ADRB3
SCHEMBL11748971 0.77 ADRB2 (0.64) MEN1KMT2AADRB1CYP2D6KCNH2
SCHEMBL11751622 0.76 ADRB2 (0.56) MEN1KMT2AADRB1CYP2D6SLC6A2
SCHEMBL11237234 0.76 CYP2D6 (0.71) CA2MEN1HTTKMT2AADRB1
Hydrochloric Acid SCHEMBL11749004 0.76 ADRB2 (0.55) MEN1KMT2AADRB1CYP2D6ADRB2
SCHEMBL21950993 0.75 CA9 (0.59) CA2MEN1KMT2ACYP2D6CA12
SCHEMBL28669393 0.74 MEN1 (0.47) CA2MEN1HTTKMT2AADRB1
SCHEMBL11751396 0.74 MEN1 (0.47) CA2MEN1HTTKMT2AADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4056626-A ADRENERGIC BLOCKING AGENTS KAKENYAKU KAKO CO., LTD. (JA) 1977-11-01 US claimed
US-4056626-A ADRENERGIC BLOCKING AGENTS KAKENYAKU KAKO CO., LTD. (JA) 1977-11-01 US disclosed