SCHEMBL11754347

SCHEMBL11754347

C#CCOC(=O)C1=C(C)N(C)C(C)=C(C(=O)OCC#C)C1c1ccccc1[N+](=O)[O-]

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.49
CACNA1C Q13936 4/20 0.49
CACNA1D Q01668 4/20 0.49
CACNA1F O60840 3/20 0.49
CACNA1S Q13698 3/20 0.49
ADORA3 P0DMS8 3/20 0.49
LMNA P02545 3/20 0.49
CYP1A2 P05177 3/20 0.49
KDM4E B2RXH2 3/20 0.49
MAPT P10636 3/20 0.49
ABCC4 O15439 2/20 0.49
ABCB11 O95342 2/20 0.49
ADORA2A P29274 2/20 0.49
ADORA1 P30542 2/20 0.49
OPRM1 P35372 2/20 0.49
SCN1A P35498 2/20 0.49
HTR2B P41595 2/20 0.49
KCNH2 Q12809 2/20 0.49
SCN5A Q14524 2/20 0.49
SCN2A Q99250 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11748298 0.85 CACNA1D (0.69) TSHRCACNA1CCACNA1DCACNA1FCACNA1S
SCHEMBL11748826 0.82 CACNA1B (0.52) TSHRCACNA1CCACNA1DCACNA1FCACNA1S
SCHEMBL1672208 0.82 TSHR (0.70) TSHRCACNA1CCACNA1DCACNA1FCACNA1S
SCHEMBL11827679 0.82 CYP1A2 (0.77) TSHRCACNA1CCACNA1DCACNA1FCACNA1S
SCHEMBL11754353 0.81 CACNA1C (0.43) TSHRCACNA1CCACNA1DCACNA1FCACNA1S
SCHEMBL10733629 0.80 CACNA1F (0.76) TSHRCACNA1CCACNA1DCACNA1FCACNA1S
SCHEMBL11447102 0.80 TSHR (0.57) TSHRCACNA1CCACNA1DCACNA1FCACNA1S
SCHEMBL11742384 0.80 ADORA3 (0.57) TSHRCACNA1CCACNA1DCACNA1FCACNA1S
SCHEMBL4608919 0.80 CACNA1C (0.64) TSHRCACNA1CCACNA1DCACNA1FCACNA1S
SCHEMBL11749142 0.80 NPSR1 (0.51) TSHRCACNA1CCACNA1DCACNA1FCACNA1S

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4048171-A 1,4-Dihydropyridines BAYER AKTIENGESELLSCHAFT (DT) 1977-09-13 US claimed
US-4048171-A 1,4-Dihydropyridines BAYER AKTIENGESELLSCHAFT (DT) 1977-09-13 US disclosed