SCHEMBL11754353

SCHEMBL11754353

C#CCCC#COC(=O)C1=C(C)N(C)C(C)=C(C(=O)O)C1c1ccccc1[N+](=O)[O-]

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 4/20 0.43
TSHR P16473 3/20 0.43
ADORA3 P0DMS8 3/20 0.43
CACNA1F O60840 3/20 0.43
CACNA1D Q01668 3/20 0.43
CACNA1S Q13698 3/20 0.43
KDM4E B2RXH2 3/20 0.43
MAPT P10636 3/20 0.43
ALDH1A1 P00352 3/20 0.43
CACNA1B Q00975 2/20 0.43
ABCC4 O15439 2/20 0.43
ABCB11 O95342 2/20 0.43
LMNA P02545 2/20 0.43
CYP1A2 P05177 2/20 0.43
ADORA2A P29274 2/20 0.43
ADORA1 P30542 2/20 0.43
OPRM1 P35372 2/20 0.43
SCN1A P35498 2/20 0.43
HTR2B P41595 2/20 0.43
KCNH2 Q12809 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11748301 0.85 ADORA3 (0.60) CACNA1CTSHRADORA3CACNA1FCACNA1D
SCHEMBL11752019 0.83 POLB (0.34) TSHRKDM4EMAPTCACNA1BLMNA
SCHEMBL11749151 0.82 KDM4E (0.41) TSHRADORA3KDM4EMAPTCACNA1B
SCHEMBL11683170 0.81 TSHR (0.65) CACNA1CTSHRADORA3CACNA1FCACNA1D
SCHEMBL11754347 0.81 TSHR (0.49) CACNA1CTSHRADORA3CACNA1FCACNA1D
SCHEMBL11752310 0.78 ALDH1A1 (0.57) TSHRKDM4EMAPTALDH1A1TP53
SCHEMBL4608919 0.78 CACNA1C (0.64) CACNA1CTSHRADORA3CACNA1FCACNA1D
SCHEMBL1672208 0.77 TSHR (0.70) CACNA1CTSHRADORA3CACNA1FCACNA1D
SCHEMBL11780568 0.74 CACNA1B (0.46) CACNA1CTSHRADORA3CACNA1FCACNA1D
SCHEMBL11752128 0.74 KDM4E (0.41) CACNA1CTSHRCACNA1FCACNA1DCACNA1S

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4048171-A 1,4-Dihydropyridines BAYER AKTIENGESELLSCHAFT (DT) 1977-09-13 US claimed
US-4048171-A 1,4-Dihydropyridines BAYER AKTIENGESELLSCHAFT (DT) 1977-09-13 US disclosed