SCHEMBL11782822

SCHEMBL11782822

COc1ccc2c(C3=CCN(Cc4ccccc4)CC3)c(C)[nH]c2c1

nearest known ligand 0.67

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 3/20 0.67
HTR1A P08908 10/20 0.62
DRD2 P14416 10/20 0.62
HTR2A P28223 2/20 0.53
ACHE P22303 1/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
KDM4E B2RXH2 2/20 0.48
ALDH1A1 P00352 2/20 0.48
POLB P06746 1/20 0.48
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11785343 0.90 DRD2 (0.62) HTR6HTR1ADRD2HTR2AACHE
SCHEMBL11637132 0.85 HTR6 (0.78) HTR6HTR1ADRD2HTR2AACHE
SCHEMBL11315770 0.84 HTR6 (0.64) HTR6HTR1ADRD2
Hydrochloric Acid SCHEMBL11639446 0.84 HTR6 (0.76) HTR6HTR1ADRD2HTR2AACHE
Hydrochloric Acid SCHEMBL11318655 0.83 HTR6 (0.62) HTR6HTR1ADRD2
SCHEMBL11786344 0.80 HTR1A (0.85) HTR1ADRD2HTR2A
SCHEMBL4194997 0.76 HTR1A (1.00) HTR1ADRD2HTR2AACHE
SCHEMBL238334 0.76 MEN1 (0.66) HTR1ADRD2HTR2AMEN1KMT2A
Hydrochloric Acid SCHEMBL19066024 0.75 MEN1 (0.65) HTR1ADRD2HTR2AMEN1KMT2A
SCHEMBL7969931 0.75 MEN1 (0.65) HTR1ADRD2HTR2AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3988453-A Novel phenothiazines as neuroleptics ROUSSEL-UCLAF (FR) 1976-10-26 US disclosed
US-3950527-A SEDATIVES ROUSSEL-UCLAF (FR) 1976-04-13 US disclosed
US-3947578-A Omega-[4-(3\"-indolyl)-piperidino]-alkyl-arylketones as nevroleptics ROUSSEL UCLAF (FR) 1976-03-30 US disclosed