SCHEMBL11800981

SCHEMBL11800981

CCOc1c(C(=O)O)sc2ccc(Br)cc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 1/20 0.46
CA12 O43570 1/20 0.44
CA9 Q16790 1/20 0.44
PTPN1 P18031 4/20 0.40
PTPN2 P17706 3/20 0.40
EPM2A O95278 1/20 0.40
PTPN22 Q9Y2R2 1/20 0.40
GPR35 Q9HC97 1/20 0.39
THRB P10828 1/20 0.39
AKR1C2 P52895 1/20 0.39
AKR1C1 Q04828 1/20 0.39
SENP5 Q96HI0 2/20 0.39
SENP2 Q9HC62 2/20 0.39
SENP1 Q9P0U3 2/20 0.39
PRNP P04156 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
PPARG P37231 1/20 0.38
HIF1A Q16665 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17173230 0.84 MCL1 (0.48) EDNRAPTPN1PTPN2GPR35SENP5
SCHEMBL6995489 0.83 EDNRA (0.54) EDNRAPTPN1PRNPCYP1A2PPARG
SCHEMBL15697543 0.81 EDNRA (0.44) EDNRAPTPN1PTPN2SENP5SENP2
SCHEMBL15697532 0.80 PTPN2 (0.56) EDNRAPTPN1PTPN2SENP5SENP2
SCHEMBL11799095 0.79 SENP5 (0.44) EDNRASENP5SENP2SENP1CYP1A2
SCHEMBL11794869 0.76 ICAM1 (0.38) CA12CA9NPSR1RXFP1SMN1; SMN2
SCHEMBL11794862 0.76 GLA (0.53) CYP1A2CYP2C9NPSR1ALDH1A1SMN1; SMN2
SCHEMBL2896475 0.76 GPR35 (0.58) PTPN1PTPN2EPM2APTPN22GPR35
SCHEMBL20563613 0.76 MCL1 (0.60) PTPN1PTPN2EPM2APTPN22GPR35
Bromomethane SCHEMBL11883047 0.75 ICAM1 (0.37) CA12CA9SENP5SENP2SENP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3976780-A Methods of protection against emesis in mammals by administration of a 3-alkoxy-thianaphthene-2-carboxamide SOCIETE D'ETUDES SCIENTIFIQUES ET INDUSTRIELLES L'ILE-DE-FRANCE (FR) 1976-08-24 US disclosed
US-3954748-A ANTIEMETICS SOCIETE D'ETUDES SCIENTIFIQUES ET INDUSTRIELLES DE L'ILE-DE-FRANCE (FR) 1976-05-04 US disclosed