SCHEMBL11883102

SCHEMBL11883102

NC(=O)n1nc2ccccc2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.40
KDM4E B2RXH2 4/20 0.39
HPGD P15428 2/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
MAPT P10636 3/20 0.38
ALDH1A1 P00352 3/20 0.38
TSHR P16473 2/20 0.38
LMNA P02545 2/20 0.38
SCN4A P35499 2/20 0.38
MAPK1 P28482 1/20 0.38
SCN5A Q14524 1/20 0.38
SCN9A Q15858 1/20 0.38
IKBKB O14920 1/20 0.37
LCK P06239 1/20 0.37
MAP2K3 P46734 1/20 0.37
MAP2K6 P52564 1/20 0.37
BTK Q06187 1/20 0.37
MAP3K19 Q56UN5 1/20 0.37
NEK10 Q6ZWH5 1/20 0.37
HSD17B10 Q99714 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL523395 0.78 HPGD (0.46) PARP1KDM4EHPGDSMN1; SMN2MAPT
SCHEMBL8143932 0.76 NPC1 (0.44) KDM4EHPGDSMN1; SMN2MAPTALDH1A1
SCHEMBL8156271 0.73 HPGD (0.50) KDM4EHPGDSMN1; SMN2MAPTALDH1A1
SCHEMBL3689757 0.71 KDM4E (0.40) PARP1KDM4EHPGDSMN1; SMN2MAPT
SCHEMBL11751025 0.71 ALDH1A1 (0.50) SMN1; SMN2ALDH1A1BCHEACHEKMT2A
SCHEMBL31707307 0.71 HPGD (0.40) PARP1KDM4EHPGDSMN1; SMN2MAPT
SCHEMBL103176 0.71 KDM4E (0.55) KDM4EHPGDSMN1; SMN2MAPTALDH1A1
SCHEMBL20818702 0.70 DGAT1 (0.43) KDM4EHPGDSMN1; SMN2MAPTALDH1A1
Water SCHEMBL994995 0.69 KDM4E (0.52) KDM4EHPGDSMN1; SMN2MAPTALDH1A1
Ammonia Solution, Strong SCHEMBL2472975 0.69 KDM4E (0.52) KDM4EHPGDSMN1; SMN2MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2668157-A1 PROTEASE ACTIVATED RECEPTOR 2 (PAR2) ANTAGONISTS Proximagen Limited (GB) 2013-12-04 EP disclosed
WO-2012101453-A1 PROTEASE ACTIVATED RECEPTOR 2 (PAR2) ANTAGONISTS PROXIMAGEN LTD. (GB) 2012-08-02 WO disclosed
US-3915979-A Preparation of benzotriazole-2-carboxamides SMITHKLINE BECKMAN CORPORATION 1975-10-28 US disclosed
US-3915979-A Preparation of benzotriazole-2-carboxamides SMITHKLINE BECKMAN CORPORATION 1975-10-28 US disclosed