SCHEMBL1189327

SCHEMBL1189327

Cc1cc(NN)nnc1Cl

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.43
GAA P10253 4/20 0.43
ALDH1A1 P00352 3/20 0.43
EDNRA P25101 1/20 0.38
GOT1 P17174 2/20 0.34
KDM4E B2RXH2 3/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
BRD4 O60885 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
LMNA P02545 1/20 0.32
PKM P14618 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrazine SCHEMBL3661754 0.96 ALDH1A1 (0.41) MAPTGAAALDH1A1EDNRAGOT1
Bromide SCHEMBL3811129 0.78 ALDH1A1 (0.31) ALDH1A1
SCHEMBL11822056 0.76 TDP1 (0.54) MAPTGAAALDH1A1GOT1KDM4E
SCHEMBL11833039 0.75 GAA (0.41) MAPTGAAALDH1A1GOT1KDM4E
SCHEMBL31226082 0.75 GAA (0.41) MAPTGAAALDH1A1GOT1KDM4E
SCHEMBL992666 0.75 GAA (0.41) MAPTGAAALDH1A1GOT1KDM4E
SCHEMBL9907139 0.74 GAA (0.39) MAPTGAAALDH1A1GOT1KDM4E
SCHEMBL2646767 0.74 GAA (0.39) MAPTGAAALDH1A1GOT1KDM4E
SCHEMBL1189496 0.74 GAA (0.39) MAPTGAAALDH1A1GOT1KDM4E
SCHEMBL11632340 0.72 L3MBTL1 (0.46) MAPTALDH1A1EDNRASMN1; SMN2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 94 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250376475-A1 ION CHANNEL MODULATORS PRAXIS PREC MEDICINES INC (US) 2025-12-11 US disclosed
US-12312333-B2 SK channel positive allosteric modulators CHAPMAN UNIVERSITY (US) 2025-05-27 US disclosed
CN-119371426-A Ion channel modulators 普拉克西斯精密药物股份有限公司 2025-01-28 CN disclosed
CN-119350320-A Ion channel modulators 普拉克西斯精密药物股份有限公司 2025-01-24 CN disclosed
EP-4487916-A2 ION CHANNEL MODULATORS Praxis Precision Medicines, Inc. (US) 2025-01-08 EP disclosed
US-20240317705-A1 POTASSIUM CHANNEL MODULATORS NOVARTIS AG (CH) 2024-09-26 US disclosed
US-20240132501-A1 ION CHANNEL MODULATORS PRAXIS PRECISION MEDICINES, INC. (US) 2024-04-25 US disclosed
CN-117756800-A Ion channel modulators 普拉克西斯精密药物股份有限公司 2024-03-26 CN disclosed
US-11866439-B2 Ion channel modulators PRAXIS PRECISION MEDICINES, INC. (US) 2024-01-09 US disclosed
US-11731978-B2 3-(ethoxydifluoromethyl)-6-(5-fluoro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl)-[1,2,4]triazolo[4,3-a]pyridine as an ion channel modulator PRAXIS PRECISION MEDICINES, INC. (US) 2023-08-22 US disclosed
US-20090312333-A1 2-Oxo-1-Pyrrolidine Derivatives, Processes for Preparing Them and Their Uses UCB PHARMA, S.A. (BE) 2009-12-17 US disclosed
WO-2009097971-A1 TRIAZOLIUM SALTS AS PAR1 INHIBITORS, PRODUCTION THEREOF, AND USE AS MEDICAMENTS SANOFI-AVENTIS (FR) 2009-08-13 WO disclosed
WO-2009097970-A1 TRIAZOLOPYRIDAZINES AS PAR1 INHIBITORS, PRODUCTION THEREOF, AND USE AS MEDICAMENTS SANOFI-AVENTIS (FR) 2009-08-13 WO disclosed
WO-2009081197-A1 BICYCLIC DERIVATIVES FOR USE IN THE TREATMENT OF ANDROGEN RECEPTOR ASSOCIATED CONDITIONS ASTRAZENECA AB (SE) 2009-07-02 WO disclosed
US-20090156607-A1 2-OXO-1-PYRROLIDINE DERIVATIVES UCB, S.A. (BE) 2009-06-18 US disclosed
US-20090156607-A1 2-OXO-1-PYRROLIDINE DERIVATIVES UCB, S.A. (BE) 2009-06-18 US disclosed
US-4578464-A 6-Hydroxyalkylamino-8-methyl-1,2,4-triazolo-[4,3-b]pyridazine and related compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1986-03-25 US disclosed
EP-0029130-B1 3,6,7,8-SUBSTITUTED-S-TRIAZOLO(4,3-B)-PYRIDAZINES, THEIR PREPARATION AND COMPOSITIONS COMPRISING THEM THE DOW CHEMICAL COMPANY (US) 1985-12-04 EP disclosed
US-4526890-A Respiratory system disorders THE DOW CHEMICAL COMPANY (US) 1985-07-02 US disclosed
EP-0029130-A1 3,6,7,8-Substituted-s-triazolo(4,3-b)-pyridazines, their preparation and compositions comprising them THE DOW CHEMICAL COMPANY (US) 1981-05-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11731978-B2 3-(ethoxydifluoromethyl)-6-(5-fluoro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl)-[1,2,4]triazolo[4,3-a]pyridine as an ion channel modulator SCN1A, SCN3A, CACNA1F MAPT 692/4885GAA 3450/4885ALDH1A1 1904/4885
US-20240132501-A1 ION CHANNEL MODULATORS SCN1A, SCN3A, SCN2A MAPT 662/4885GAA 2007/4885ALDH1A1 1953/4885
US-20240317705-A1 POTASSIUM CHANNEL MODULATORS KCNJ11, KCNJ2, KCNJ1 MAPT 2009/4885GAA 1172/4885ALDH1A1 1320/4885
US-11866439-B2 Ion channel modulators SCN1A, SCN3A, SCN2A MAPT 662/4885GAA 2007/4885ALDH1A1 1953/4885
US-20090312333-A1 2-Oxo-1-Pyrrolidine Derivatives, Processes for Preparing Them and Their Uses CYP3A4, CYP1B1, CYP2D6 MAPT 2583/4885GAA 138/4885ALDH1A1 560/4885
US-12312333-B2 SK channel positive allosteric modulators KCNN1, KCNN4, KCNN2 MAPT 2936/4885GAA 2648/4885ALDH1A1 4418/4885
US-20090156607-A1 2-OXO-1-PYRROLIDINE DERIVATIVES OPRD1, PPOX, CYP2D6 MAPT 1512/4885GAA 255/4885ALDH1A1 447/4885
US-20250376475-A1 ION CHANNEL MODULATORS SCN1A, SCN3A, SCN2A MAPT 662/4885GAA 2007/4885ALDH1A1 1953/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.