SCHEMBL11903463

SCHEMBL11903463

FC(F)(F)Oc1ccc2[nH]c(-c3cccnc3)nc2c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.61
MAPT P10636 3/20 0.61
RAB9A P51151 3/20 0.61
NPC1 O15118 2/20 0.61
ALDH1A1 P00352 2/20 0.61
HPGD P15428 2/20 0.61
STAT1 P42224 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
NPY5R Q15761 2/20 0.57
LDHA P00338 1/20 0.57
EPHX2 P34913 1/20 0.57
CYP11B1 P15538 3/20 0.54
KIT P10721 1/20 0.53
DGAT1 O75907 1/20 0.52
KCNH2 Q12809 1/20 0.52
HTT P42858 2/20 0.51
CBFB Q13951 3/20 0.51
RUNX1 Q01196 4/20 0.49
TRPV1 Q8NER1 1/20 0.49
IDO1 P14902 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11903458 0.90 CYP11B1 (0.64) KDM4EMAPTRAB9ANPC1ALDH1A1
SCHEMBL11903477 0.85 TRPV1 (0.57) KDM4EMAPTRAB9ANPC1ALDH1A1
SCHEMBL19970729 0.82 NAMPT (0.49) KDM4EMAPTRAB9ANPC1ALDH1A1
SCHEMBL4036018 0.81 KIT (0.49) KDM4EMAPTRAB9ANPC1ALDH1A1
SCHEMBL19970839 0.81 KIT (0.49) KDM4EMAPTRAB9ANPC1ALDH1A1
SCHEMBL5683118 0.81 DGAT1 (0.73) KDM4EMAPTRAB9ANPC1ALDH1A1
SCHEMBL11903464 0.79 TRPV1 (0.60) KDM4ERAB9ANPC1ALDH1A1SMN1; SMN2
SCHEMBL11903487 0.79 CYP1A2 (0.54) KDM4ERAB9ANPC1ALDH1A1HPGD
SCHEMBL10175464 0.79 CYP11B1 (0.79) KDM4EMAPTRAB9ANPC1ALDH1A1
SCHEMBL11903647 0.78 TRPV1 (0.62) KDM4EMAPTRAB9ANPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8293780-B1 Anti-cancer agents based on 6-trifluoromethoxybenzimidazole derivatives and method of making U.S. DEPARTMENT OF ENERGY (US) 2012-10-23 US disclosed
US-8242284-B1 Anti-cancer agents based on 6-trifluoromethoxybenzimidazole derivatives and method of making THE UNITED STATES OF AMERICA AS REPRESENTED BY THE UNITED STATES DEPARTMENT OF ENERGY (US) 2012-08-14 US disclosed