SCHEMBL11903515

SCHEMBL11903515

CC(C)c1ccc(-c2nc3cc(OC(F)(F)F)ccc3[nH]2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 3/20 0.58
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
CHEK2 O96017 1/20 0.44
RUNX1 Q01196 4/20 0.44
CBFB Q13951 3/20 0.44
DHODH Q02127 1/20 0.43
NPC1 O15118 2/20 0.43
ALDH1A1 P00352 2/20 0.43
PKM P14618 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 1/20 0.43
RAB9A P51151 1/20 0.43
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11903519 0.90 TRPV1 (0.72) TRPV1HDAC3HDAC1HDAC2HDAC8
SCHEMBL11903494 0.86 TRPV1 (0.62) TRPV1CHEK2RUNX1CBFBNPC1
SCHEMBL11903440 0.86 TRPV1 (0.58) TRPV1CHEK2RUNX1CBFBDHODH
SCHEMBL11903647 0.86 TRPV1 (0.62) TRPV1CHEK2RUNX1CBFBNPC1
SCHEMBL11903467 0.85 TRPV1 (0.57) TRPV1HDAC3HDAC1HDAC2HDAC8
SCHEMBL11903464 0.84 TRPV1 (0.60) TRPV1CHEK2RUNX1CBFBDHODH
SCHEMBL11903477 0.83 TRPV1 (0.57) TRPV1CHEK2RUNX1CBFBDHODH
SCHEMBL11903531 0.82 TRPV1 (0.58) TRPV1CHEK2RUNX1CBFBDHODH
SCHEMBL11903644 0.81 TRPV1 (0.56) TRPV1CHEK2RUNX1CBFBNPC1
SCHEMBL13305849 0.80 TRPV1 (0.55) TRPV1HDAC3HDAC1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8293780-B1 Anti-cancer agents based on 6-trifluoromethoxybenzimidazole derivatives and method of making U.S. DEPARTMENT OF ENERGY (US) 2012-10-23 US disclosed
US-8242284-B1 Anti-cancer agents based on 6-trifluoromethoxybenzimidazole derivatives and method of making THE UNITED STATES OF AMERICA AS REPRESENTED BY THE UNITED STATES DEPARTMENT OF ENERGY (US) 2012-08-14 US disclosed