SCHEMBL11903531

SCHEMBL11903531

CSc1ccc(-c2nc3cc(OC(F)(F)F)ccc3[nH]2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 3/20 0.58
CHEK2 O96017 2/20 0.52
RUNX1 Q01196 5/20 0.44
CBFB Q13951 3/20 0.44
NPC1 O15118 2/20 0.43
ALDH1A1 P00352 2/20 0.43
PKM P14618 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 1/20 0.43
RAB9A P51151 1/20 0.43
DHODH Q02127 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11903647 0.86 TRPV1 (0.62) TRPV1CHEK2RUNX1CBFBNPC1
SCHEMBL11903494 0.86 TRPV1 (0.62) TRPV1CHEK2RUNX1CBFBNPC1
SCHEMBL11903464 0.84 TRPV1 (0.60) TRPV1CHEK2RUNX1CBFBNPC1
SCHEMBL11903440 0.83 TRPV1 (0.58) TRPV1CHEK2RUNX1CBFBNPC1
SCHEMBL11903477 0.83 TRPV1 (0.57) TRPV1CHEK2RUNX1CBFBNPC1
SCHEMBL11903515 0.82 TRPV1 (0.58) TRPV1CHEK2RUNX1CBFBNPC1
SCHEMBL11903467 0.82 TRPV1 (0.57) TRPV1CHEK2RUNX1CBFBNPC1
SCHEMBL10766038 0.81 NPBWR1 (0.58) NPC1KDM4ERAB9APOLBNPBWR1
SCHEMBL11903644 0.81 TRPV1 (0.56) TRPV1CHEK2RUNX1CBFBNPC1
SCHEMBL13305849 0.80 TRPV1 (0.55) TRPV1CHEK2RUNX1CBFB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8293780-B1 Anti-cancer agents based on 6-trifluoromethoxybenzimidazole derivatives and method of making U.S. DEPARTMENT OF ENERGY (US) 2012-10-23 US disclosed
US-8242284-B1 Anti-cancer agents based on 6-trifluoromethoxybenzimidazole derivatives and method of making THE UNITED STATES OF AMERICA AS REPRESENTED BY THE UNITED STATES DEPARTMENT OF ENERGY (US) 2012-08-14 US disclosed