SCHEMBL11904550

SCHEMBL11904550

Cc1ccc(S(=O)(=O)Oc2cc(C(F)(F)F)nc3c(C(F)(F)F)cccc23)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.47
ESR1 P03372 1/20 0.47
GAA P10253 1/20 0.47
KMT2A Q03164 1/20 0.47
ESR2 Q92731 1/20 0.47
SLC2A1 P11166 1/20 0.41
SDHB P21912 2/20 0.41
CYP1A2 P05177 2/20 0.40
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
NR1H2 P55055 2/20 0.38
CYP2D6 P10635 2/20 0.38
PTGS2 P35354 2/20 0.38
PTGS1 P23219 1/20 0.38
ADORA2A P29274 5/20 0.38
ADORA1 P30542 5/20 0.38
KCNH2 Q12809 4/20 0.38
CYP3A4 P08684 3/20 0.38
ADORA3 P0DMS8 2/20 0.38
LMNA P02545 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11904341 0.83 SLC2A1 (0.42) MEN1ESR1KMT2ASLC2A1SDHB
SCHEMBL7071544 0.76 LMNA (0.52) MEN1ESR1GAAKMT2AESR2
SCHEMBL9872956 0.75 GAA (0.46) MEN1ESR1GAAKMT2AESR2
SCHEMBL11166946 0.74 CYP2D6 (0.43) MEN1ESR1KMT2ASLC2A1CYP1A2
SCHEMBL2790280 0.72 ALDH1A1 (0.48) ESR1CYP1A2NR1H2CYP2D6PTGS2
SCHEMBL1655812 0.70 KCNH2 (0.49) ESR1SLC2A1CYP1A2CYP2D6PTGS2
SCHEMBL6938149 0.70 MEN1 (0.57) MEN1ESR1GAAKMT2AESR2
SCHEMBL10698356 0.70 CYP1A2 (0.41) MEN1ESR1GAAKMT2AESR2
SCHEMBL1073454 0.69 MEN1 (0.68) MEN1ESR1GAAKMT2AESR2
SCHEMBL3843866 0.69 LMNA (0.50) MEN1ESR1GAAKMT2AESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012107532-A1 4-AMINOALCOHOLQUINOLINE DERIVATIVES, ENANTIOSELECTIVE SYNTHESIS METHODS AND THE USE THEREOF Université de Picardie Jules Verne (FR) 2012-08-16 WO disclosed
EP-2487157-A1 Enantioselective synthesis method of 4-aminoalcoholquinoline derivatives and the use Université de Picardie Jules Verne (FR) 2012-08-15 EP disclosed