SCHEMBL11939409

SCHEMBL11939409

c1ccc(CN2Cc3ccccc3C3(CCN(C4CCNCC4)CC3)C2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 12/20 0.48
TSHR P16473 3/20 0.48
CYP2C19 P33261 3/20 0.48
CYP2D6 P10635 3/20 0.48
TP53 P04637 2/20 0.48
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
ALDH1A1 P00352 2/20 0.48
CYP2C9 P11712 2/20 0.48
DRD2 P14416 1/20 0.46
NFKB1 P19838 1/20 0.46
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
MAPK1 P28482 1/20 0.46
HTR2B P41595 1/20 0.46
MTOR P42345 1/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
BLM P54132 1/20 0.46
PMP22 Q01453 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11939778 0.82 OPRM1 (0.42) SIGMAR1OPRM1OPRK1OPRL1SLC18A3
SCHEMBL12934948 0.79 ALDH1A1 (0.49) SIGMAR1ALDH1A1MEN1KMT2AOPRM1
SCHEMBL11939435 0.78 OPRM1 (0.40) SIGMAR1HTR2AHTR2CHTR2BOPRM1
SCHEMBL24481541 0.77 SIGMAR1 (0.60) SIGMAR1TSHRCYP2C19CYP2D6TP53
SCHEMBL14467581 0.76 SIGMAR1 (0.58) SIGMAR1TSHRCYP2C19CYP2D6TP53
SCHEMBL11939412 0.76 KCNH2 (0.41) SIGMAR1HTR2AHTR2CHTR2BOPRM1
SCHEMBL1206722 0.75 SIGMAR1 (0.64) SIGMAR1TSHRCYP2C19ALDH1A1CYP2C9
SCHEMBL11940836 0.74 NAMPT (0.40) HTR2AHTR2CHTR2BOPRM1OPRK1
SCHEMBL11939419 0.73 OPRM1 (0.42) SIGMAR1HTR2AHTR2CHTR2BKMT2A
SCHEMBL11939156 0.73 KEAP1 (0.46) SIGMAR1HTR2AHTR2CHTR2BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817036-B1 MODULATORS OF MUSCARINIC RECEPTORS VERTEX PHARMA (US) 2012-07-04 EP disclosed