Timobesone Acetate

Timobesone Acetate

SCHEMBL119875

CSC(=O)[C@@]1(OC(C)=O)[C@@H](C)C[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@@]21C

nearest known ligand 0.67

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
▸ NR3C1 P04150 12/20 0.67
▸ CYP3A4 P08684 5/20 0.67
▸ PGR P06401 4/20 0.67
▸ USP2 O75604 3/20 0.67
▸ LMNA P02545 3/20 0.67
▸ NR1I2 O75469 2/20 0.67
▸ MAPT P10636 2/20 0.67
▸ SMN1; SMN2 Q16637 2/20 0.67
▸ CYP2C9 P11712 2/20 0.67
▸ MLNR O43193 1/20 0.67
▸ ABCB11 O95342 1/20 0.67
▸ CYP3A5 P20815 1/20 0.67
▸ PPARG P37231 1/20 0.67
▸ NPSR1 Q6W5P4 1/20 0.67
▸ CYP2D6 P10635 1/20 0.67
▸ MMP1 P03956 6/20 0.66
▸ ADORA3 P0DMS8 1/20 0.66
▸ DRD2 P14416 1/20 0.66
▸ OPRD1 P41143 1/20 0.66
▸ MEN1 O00255 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8859709 0.92 NR3C1 (0.74) NR3C1CYP3A4PGRUSP2LMNA
SCHEMBL11229266 0.91 NR3C1 (0.66) NR3C1CYP3A4PGRUSP2LMNA
SCHEMBL11223809 0.90 NR3C1 (0.70) NR3C1CYP3A4PGRUSP2LMNA
SCHEMBL11228765 0.90 NR3C1 (0.69) NR3C1CYP3A4PGRUSP2LMNA
SCHEMBL11689579 0.89 NR3C1 (0.69) NR3C1CYP3A4PGRUSP2LMNA
SCHEMBL11246943 0.89 NR3C1 (0.69) NR3C1CYP3A4PGRUSP2LMNA
SCHEMBL11813525 0.89 NR3C1 (0.69) NR3C1CYP3A4PGRUSP2LMNA
SCHEMBL11228768 0.89 NR3C1 (0.69) NR3C1CYP3A4PGRUSP2LMNA
SCHEMBL11690649 0.89 NR3C1 (0.69) NR3C1CYP3A4PGRUSP2LMNA
SCHEMBL6986508 0.88 NR3C1 (0.83) NR3C1CYP3A4PGRUSP2MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 292 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024189434-A1 USE OF NADOLOL TO TREAT PULMONARY SYMPTOMS ASSOCIATED WITH INFECTIONS WITH SARS-CoV-2 CHRONIC AIRWAY THERAPEUTICS LIMITED (AU) 2024-09-19 — — WO claimed
US-20220096498-A1 INJECTABLE SUSTAINED-RELEASE FORMULATIONS FOR TREATMENT OF JOINT PAIN AND INFLAMMATION FORDOZ PHARMA CORP. (US) 2022-03-31 — — US claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 — — US claimed
US-8268352-B2 Modified release composition for highly soluble drugs TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-18 — — US claimed
US-8263125-B2 Dosage form for high dose-high solubility active ingredients that provides for immediate release and modified release of the active ingredients TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-11 — — US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 — — US claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 — — EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 — — WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 — — US claimed
US-20060024365-A1 Novel dosage form VAYA NAVIN 2006-02-02 — — US claimed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 — — US claimed
US-20060018934-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 — — US claimed
US-5145675-A Polymerizing suspended monomers in presence of porogen to form rigid crosslinked beads with internal pore network, extracting porogen, introducing active substance ADVANCED POLYMER SYSTEMS, INC. (US) 1992-09-08 — — US claimed
US-20260124244-A1 MEGAKARYOCYTE DERIVATIVES FOR TREATMENT OF DRY EYE DISEASES STELLULAR BIO, INC. (US) 2026-05-07 — — US disclosed
US-12589102-B2 Injectable sustained-release formulations for treatment of joint pain and inflammation FORDOZ PHARMA CORP. (US) 2026-03-31 — — US disclosed
EP-4706683-A2 CHEWABLE FORMULATIONS Elanco Tiergesundheit AG (CH) 2026-03-11 — — EP disclosed
US-4962133-A PRECIPITATION POLYMERIZATION; CONTROLLING PARTICLE SIZE BY VARYING RATE OF STIRRING DOW CORNING CORPORATION (US) 1990-10-09 — — US disclosed
EP-0277211-A4 POLYMERIC CARRIER COMPOSITIONS AND METHODS FOR THEIR PREPARATION AND USE — 1990-09-05 — — EP disclosed
EP-0277211-A1 POLYMERIC CARRIER COMPOSITIONS AND METHODS FOR THEIR PREPARATION AND USE. ADVANCED POLYMER SYSTEMS INC (US) 1988-08-10 — — EP disclosed
WO-1988001164-A1 POLYMERIC CARRIER COMPOSITIONS AND METHODS FOR THEIR PREPARATION AND USE ADVANCED POLYMER SYSTEMS, INC. (US) 1988-02-25 — — WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260124244-A1 MEGAKARYOCYTE DERIVATIVES FOR TREATMENT OF DRY EYE DISEASES MYH10, PDGFA, MPL NR3C1 4364/4885CYP3A4 2902/4885PGR 157/4885
US-12589102-B2 Injectable sustained-release formulations for treatment of joint pain and inflammation IL1B, TNF, MIF NR3C1 25/4885CYP3A4 1290/4885PGR 38/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.

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