Deferoxamine

Deferoxamine

SCHEMBL119983

CC(=O)N(O)CCCCCNC(=O)CCC(=O)N(O)CCCCCNC(=O)CCC(=O)N(O)CCCCCN.CS(=O)(=O)[O-].[H+]

nearest known ligand 0.91

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of Deferoxamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.91
LMNA P02545 1/20 0.91
GAA P10253 1/20 0.91
SMN1; SMN2 Q16637 1/20 0.91
KDM4A O75164 9/20 0.84
HIF1A Q16665 1/20 0.84
TET2 Q6N021 1/20 0.84
DOHH Q9BU89 1/20 0.84
PAOX Q6QHF9 2/20 0.39
SLC6A5 Q9Y345 2/20 0.38
KDM4C Q9H3R0 8/20 0.35
CASP2 P42575 1/20 0.33
KDM5A P29375 1/20 0.32
KDM7A Q6ZMT4 1/20 0.32
PHF8 Q9UPP1 1/20 0.32
KDM2A Q9Y2K7 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Deferoxamine SCHEMBL10579133 0.98 KDM4E (0.91) KDM4ELMNAGAASMN1; SMN2KDM4A
Deferoxamine SCHEMBL18983317 0.98 KDM4E (0.91) KDM4ELMNAGAASMN1; SMN2KDM4A
Deferoxamine SCHEMBL1699778 0.95 KDM4E (1.00) KDM4ELMNAGAASMN1; SMN2KDM4A
Deferoxamine SCHEMBL119982 0.95 KDM4E (1.00) KDM4ELMNAGAASMN1; SMN2KDM4A
SCHEMBL30036991 0.95 KDM4E (1.00) KDM4ELMNAGAASMN1; SMN2KDM4A
Deferoxamine SCHEMBL7715593 0.95 KDM4E (1.00) KDM4ELMNAGAASMN1; SMN2KDM4A
Deferoxamine SCHEMBL3953046 0.94 KDM4E (0.97) KDM4ELMNAGAASMN1; SMN2KDM4A
Deferoxamine SCHEMBL9351925 0.94 KDM4E (0.97) KDM4ELMNAGAASMN1; SMN2KDM4A
Deferoxamine SCHEMBL2165915 0.93 KDM4E (0.95) KDM4ELMNAGAASMN1; SMN2KDM4A
Deferoxamine SCHEMBL1034134 0.93 KDM4E (0.95) KDM4ELMNAGAASMN1; SMN2KDM4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3400 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144251-A1 ANTIMICROBIAL NANOCLAYS COMPRISING CATIONIC ANTIMICROBIALS, METHOD OF PREPARATION AND USES THEREOF POLYAMYNA NANOTECH INC. (CA) 2026-05-28 US claimed
WO-2025224448-A1 STABLE BIORELEVANT COMPOSITIONS AND MEDIA FOR IN VITRO TESTING BIORELEVANT.COM LIMITED (GB) 2025-10-30 WO claimed
US-20250332118-A1 NOVEL ORAL CARE FORMULATIONS FOR TREATMENT OF XEROSTOMIA LIVIONEX INC (US) 2025-10-30 US claimed
US-20250319214-A1 A NOVEL KIT FOR RADIOPHARMACEUTICAL PREPARATION OF A RADIOMETAL LABELED CHELATE-FUNCTIONALIZED TARGETING CONJUGATE Life Molecular Imaging Ltd. (GB) 2025-10-16 US claimed
CN-115443162-B Drug injection device, system and method 解决方案医疗公司 2025-05-06 CN claimed
US-20250064739-A1 OXAZOLIDINONE LIPOSOME COMPOSITIONS AKAGERA MEDICINES, INC. (US) 2025-02-27 US claimed
CN-119464378-A Gene editing method of neutrophils 电子科技大学 2025-02-18 CN claimed
EP-4504163-A1 NOVEL ORAL CARE FORMULATIONS FOR TREATMENT OF XEROSTOMIA Livionex, Inc. (US) 2025-02-12 EP claimed
EP-4452252-A2 OXAZOLIDINONE LIPOSOME COMPOSITIONS Akagera Medicines, Inc. (US) 2024-10-30 EP claimed
EP-4362989-A2 A NOVEL KIT FOR RADIOPHARMACEUTICAL PREPARATION OF A RADIOMETAL LABELED CHELATE-FUNCTIONALIZED TARGETING CONJUGATE Life Molecular Imaging Limited (GB) 2024-05-08 EP claimed
WO-1999036055-A1 AUTOCLAVABLE PHARMACEUTICAL COMPOSITIONS CONTAINING A CHELATING AGENT NOVARTIS AG (CH) 1999-07-22 WO claimed
US-5895786-A Method for treating viral infections NEW YORK BLOOD CENTER, INC. (US) 1999-04-20 US claimed
EP-0904075-A1 METHOD FOR TREATING VIRAL INFECTIONS THE NEW YORK BLOOD CENTER, INC. (US) 1999-03-31 EP claimed
WO-1997041855-A1 METHOD FOR TREATING VIRAL INFECTIONS NEW YORK BLOOD CENTER, INC. (US) 1997-11-13 WO claimed
EP-0436005-B1 LABELED POLYPEPTIDE DERIVATIVES SANDOZ LTD (CH) 1995-03-29 EP claimed
EP-0313630-B1 SUBSTITUTED 2-ACYLPYRIDIN-ALPHA-(N)-HETARYLHYDRAZONES AND MEDICAMENTS CONTAINING SAME DEUTSCHES AUSSÄTZIGEN HILFSWERK E.V. (DE) 1992-09-16 EP claimed
EP-0436005-A1 LABELED POLYPEPTIDE DERIVATIVES. SANDOZ LTD (CH) 1991-07-10 EP claimed
WO-1991001144-A1 LABELED POLYPEPTIDE DERIVATIVES SANDOZ LTD (CH) 1991-02-07 WO claimed
EP-0313630-A1 SUBSTITUTED 2-ACYLPYRIDIN-ALPHA-(N)-HETARYLHYDRAZONES AND MEDICAMENTS CONTAINING SAME. DEUTSCHES AUSSATZIGEN HILFSWER (DE) 1989-05-03 EP claimed
WO-1988008842-A2 SUBSTITUTED 2-ACYLPYRIDIN-alpha-(N)-HETARYLHYDRAZONES AND MEDICAMENTS CONTAINING SAME DEUTSCHES AUSSÄTZIGEN HILFSWERK E.V. (DE) 1988-11-17 WO claimed