SCHEMBL2588902

SCHEMBL2588902

Cc1ccc(CNc2nc(Nc3cccc(Cl)c3)nc3ccccc23)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 2/20 0.66
PDE5A O76074 2/20 0.59
CTNNB1 P35222 1/20 0.57
TCF7L2 Q9NQB0 1/20 0.57
LMNA P02545 4/20 0.57
MAPT P10636 4/20 0.57
MAPK1 P28482 3/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
ALDH1A1 P00352 3/20 0.57
KMT2A Q03164 3/20 0.57
NPSR1 Q6W5P4 3/20 0.57
USP2 O75604 1/20 0.57
HPGD P15428 1/20 0.57
NR2F2 P24468 1/20 0.57
NPY5R Q15761 1/20 0.56
APP P05067 1/20 0.56
SLC2A1 P11166 1/20 0.55
NTRK1 P04629 2/20 0.55
PGK1 P00558 1/20 0.55
KDM4E B2RXH2 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2588890 0.92 SOS1 (0.70) SOS1PDE5ACTNNB1TCF7L2LMNA
SCHEMBL2583209 0.92 SOS1 (0.72) SOS1PDE5ACTNNB1TCF7L2LMNA
SCHEMBL2587460 0.90 SOS1 (0.65) SOS1PDE5ALMNAMAPTMAPK1
SCHEMBL2587225 0.89 SOS1 (0.66) SOS1PDE5ACTNNB1TCF7L2LMNA
SCHEMBL2590218 0.89 SOS1 (0.66) SOS1PDE5ACTNNB1TCF7L2LMNA
SCHEMBL2592287 0.89 SOS1 (0.71) SOS1PDE5ALMNAMAPTALDH1A1
SCHEMBL2590586 0.89 SLC2A1 (0.73) SOS1PDE5ACTNNB1TCF7L2LMNA
SCHEMBL2592190 0.85 NPY5R (0.78) SOS1PDE5ALMNAMAPTMAPK1
SCHEMBL12176293 0.85 SOS1 (0.72) SOS1PDE5ALMNAMAPTMAPK1
SCHEMBL2587390 0.85 SOS1 (0.66) SOS1PDE5ALMNAMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2566480-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE California Institute of Technology (US) 2013-03-13 EP disclosed
WO-2011140527-A2 METHODS AND COMPOSITIONS FOR INHIBITION OF THE TRANSITIONAL ENDOPLASMIC RETICULUM ATPASE CALIFORNIA INSTITUTE OF TECHNOLOGY AND THE UNIVERSITY OF KANSAS (US) 2011-11-10 WO disclosed