SCHEMBL12201989

SCHEMBL12201989

O=C(COc1ccc(C(O)c2cccs2)c(Cl)c1Cl)Nc1ccc2cnccc2c1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 5/20 0.58
ROCK2 O75116 6/20 0.42
CACNA2D1 P54289 2/20 0.41
LMNA P02545 2/20 0.41
MAPK1 P28482 1/20 0.41
NPC1 O15118 1/20 0.41
GALR3 O60755 1/20 0.40
STAT3 P40763 1/20 0.40
IMPDH2 P12268 1/20 0.40
POLB P06746 2/20 0.40
NOD2 Q9HC29 1/20 0.40
PRNP P04156 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12201994 0.87 NOTUM (0.59) NOTUMROCK2CACNA2D1LMNANPC1
SCHEMBL12201980 0.84 NOTUM (0.63) NOTUMROCK2LMNAMAPK1NPC1
SCHEMBL12201990 0.81 NOTUM (0.60) NOTUMLMNAMAPK1NPC1GALR3
SCHEMBL1105179 0.77 CYP2C9 (0.57) NOTUMLMNAMAPK1NPC1GALR3
SCHEMBL12201983 0.76 NOTUM (0.83) NOTUMROCK2LMNAMAPK1NPC1
SCHEMBL12201988 0.76 NOTUM (0.66) NOTUMLMNAMAPK1NPC1IMPDH2
SCHEMBL12201981 0.76 NOTUM (0.65) NOTUMLMNAMAPK1NPC1POLB
SCHEMBL11741712 0.75 CYP2C9 (0.56) LMNA
SCHEMBL1123774 0.73 NOTUM (0.57) NOTUMLMNAMAPK1NPC1POLB
SCHEMBL12201987 0.72 NOTUM (0.65) NOTUMLMNAGALR3IMPDH2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8034943-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2011-10-11 US disclosed
US-8034943-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2011-10-11 US disclosed
US-20100137364-A1 6-Aminoisoquinoline Compounds AERIE PHARMACEUTICALS, INC. (US) 2010-06-03 US disclosed
US-20100137364-A1 6-Aminoisoquinoline Compounds AERIE PHARMACEUTICALS, INC. (US) 2010-06-03 US disclosed
US-7671205-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2010-03-02 US disclosed
US-7671205-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2010-03-02 US disclosed
US-20070173530-A1 6-Aminoisoquinoline Compounds AERIE PHARMACEUTICALS, INC. (US) 2007-07-26 US disclosed
US-20070173530-A1 6-Aminoisoquinoline Compounds AERIE PHARMACEUTICALS, INC. (US) 2007-07-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100137364-A1 6-Aminoisoquinoline Compounds COQ8A, PGC, AGK NOTUM 3635/4885ROCK2 246/4885CACNA2D1 4576/4885
US-20070173530-A1 6-Aminoisoquinoline Compounds COQ8A, PGC, AGK NOTUM 3635/4885ROCK2 246/4885CACNA2D1 4576/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.