SCHEMBL12283041

SCHEMBL12283041

Cc1ccc(CCNC(=O)OC(C)(C)C)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.60
RAB9A P51151 3/20 0.60
SMN1; SMN2 Q16637 2/20 0.60
MAPT P10636 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
CA2 P00918 4/20 0.56
CA1 P00915 2/20 0.56
NAMPT P43490 1/20 0.55
PTGER4 P35408 1/20 0.51
KMT2A Q03164 2/20 0.50
GLA P06280 1/20 0.50
PLAAT3 P53816 2/20 0.49
PLAAT5 Q96KN8 2/20 0.49
PLAAT2 Q9NWW9 2/20 0.49
PLAAT4 Q9UL19 2/20 0.49
HPGD P15428 1/20 0.49
EPHX2 P34913 1/20 0.48
CNR1 P21554 1/20 0.48
NQO2 P16083 1/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL8528143 0.95 NPC1 (0.56) NPC1RAB9ASMN1; SMN2MAPTTDP1
SCHEMBL22996211 0.91 CA1 (0.54) NPC1RAB9ASMN1; SMN2MAPTTDP1
SCHEMBL27741035 0.87 CA2 (0.56) NPC1RAB9ASMN1; SMN2MAPTTDP1
SCHEMBL100146 0.87 KDM4E (0.60) NPC1RAB9ASMN1; SMN2MAPTTDP1
SCHEMBL1569661 0.87 CA2 (0.56) NPC1RAB9ASMN1; SMN2MAPTTDP1
SCHEMBL24667825 0.87 NAMPT (0.56) NPC1RAB9ASMN1; SMN2MAPTTDP1
SCHEMBL11961188 0.86 CA2 (0.55) NPC1RAB9ASMN1; SMN2MAPTTDP1
SCHEMBL1065312 0.86 CA2 (0.55) NPC1RAB9ASMN1; SMN2MAPTTDP1
SCHEMBL23449213 0.86 CA2 (0.58) MAPTTDP1CA2CA1NAMPT
SCHEMBL21521028 0.86 CA2 (0.55) NPC1RAB9ASMN1; SMN2MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115722266-A Novel aza-carbene-amido-ruthenium catalyst and preparation method and application thereof 广东药科大学 2023-03-03 CN disclosed
WO-2021106979-A1 LIQUID CRYSTAL ALIGNING AGENT, LIQUID CRYSTAL ALIGNMENT FILM, AND LIQUID CRYSTAL DISPLAY ELEMENT 日産化学株式会社 2021-06-03 WO disclosed
WO-2021041770-A1 PCSK9 ANTAGONIST COMPOUNDS MERCK SHARP & DOHME CORP. (US) 2021-03-04 WO disclosed
US-10654834-B2 Non-systemic TGR5 agonists Venenum Biodesign, LLC (US) 2020-05-19 US disclosed
US-20190330191-A1 NOVEL NON-SYSTEMIC TGR5 AGONISTS Venenum Biodesign, LLC (US) 2019-10-31 US disclosed
US-8673908-B2 Kynurenine production inhibitor KYOWA HAKKO KIRIN CO., LTD. (JP) 2014-03-18 US disclosed
US-20110237584-A1 KYNURENINE PRODUCTION INHIBITOR KYOWA KIRIN CO., LTD. (JP) 2011-09-29 US disclosed
WO-2010053182-A1 KYNURENINE PRODUCTION INHIBITOR 協和発酵キリン株式会社 (JP) 2010-05-14 WO disclosed
EP-1641465-B1 COMBINATIONS OF AN ARYL ANILINE BETA-2 ADRENERGIC RECEPTOR AGONIST AND A CORTICOSTEROID THERAVANCE INC (US) 2009-11-04 EP disclosed
CN-1293057-C Ethylenediamine derivatives DAIICHI SEIYAKU CO (JP) 2007-01-03 CN disclosed
CN-1438993-A Ethylenediamine derivatives DAIICHI SEIYAKU CO (JP) 2003-08-27 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190330191-A1 NOVEL NON-SYSTEMIC TGR5 AGONISTS GPR119, FFAR1, FFAR3 NPC1 321/4885RAB9A 3031/4885SMN1; SMN2 3965/4885
US-10654834-B2 Non-systemic TGR5 agonists GPR119, SSTR5, FFAR3 NPC1 358/4885RAB9A 3387/4885SMN1; SMN2 3817/4885
US-20110237584-A1 KYNURENINE PRODUCTION INHIBITOR KYNU, KMO, IDO1 NPC1 4522/4885RAB9A 3666/4885SMN1; SMN2 4398/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.