SCHEMBL1233669

SCHEMBL1233669

NC(=O)c1cccnc1NCCNC(=O)c1cccnc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.59
HSD17B10 Q99714 2/20 0.59
KDM4E B2RXH2 1/20 0.59
HPGD P15428 1/20 0.59
USP2 O75604 2/20 0.52
THRB P10828 1/20 0.51
RAB9A P51151 3/20 0.51
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
NPC1 O15118 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
EPHX2 P34913 3/20 0.50
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
MAPT P10636 2/20 0.48
AURKA O14965 1/20 0.48
RPS6KB1 P23443 1/20 0.48
AURKB Q96GD4 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL571346 0.82 SIRT2 (0.60) ALDH1A1HSD17B10KDM4EHPGDTHRB
SCHEMBL1233667 0.81 MAPT (0.53) ALDH1A1HSD17B10USP2THRBRAB9A
SCHEMBL25328235 0.80 THRB (0.77) ALDH1A1HSD17B10USP2THRBRAB9A
SCHEMBL7129338 0.79 KDM4E (0.63) ALDH1A1HSD17B10KDM4EHPGDRAB9A
SCHEMBL1235984 0.78 F7 (0.54) ALDH1A1HSD17B10USP2THRBRAB9A
SCHEMBL17490812 0.76 ALDH1A1 (0.75) ALDH1A1HSD17B10KDM4EHPGDRAB9A
SCHEMBL31204910 0.76 ALDH1A1 (0.58) ALDH1A1HSD17B10KDM4EHPGDUSP2
SCHEMBL3714863 0.76 ALDH1A1 (0.58) ALDH1A1HSD17B10KDM4EHPGDUSP2
SCHEMBL8351026 0.75 ALDH1A1 (0.69) ALDH1A1HSD17B10KDM4EHPGDRAB9A
SCHEMBL10725418 0.74 THRB (0.64) ALDH1A1HSD17B10USP2THRBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2285376-A1 6-AMINONICOTINAMIDE DERIVATIVES AS POTENT AND SELECTIVE HISTONE DEACETYLASE INHIBITORS Chipscreen Biosciences Ltd. (CN) 2011-02-23 EP disclosed