SCHEMBL12366183

SCHEMBL12366183

[C-]#[N+]CC(=O)NCc1cccc(Br)c1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.56
MAPT P10636 2/20 0.52
ALOX5 P09917 1/20 0.48
F10 P00742 1/20 0.47
F7 P08709 1/20 0.47
MTOR P42345 1/20 0.47
TP53 P04637 1/20 0.46
LMNA P02545 3/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HPGD P15428 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
FFAR1 O14842 1/20 0.44
FFAR4 Q5NUL3 1/20 0.44
THRB P10828 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12366093 0.82 MMP13 (0.52) NPC1TP53LMNAHPGD
SCHEMBL12366208 0.82 SRC (0.57) TP53
SCHEMBL24499495 0.81 NPC1 (0.61) NPC1MAPTALOX5F10F7
SCHEMBL6290205 0.81 NPC1 (0.61) NPC1MAPTALOX5F10F7
SCHEMBL6290206 0.81 NPC1 (0.61) NPC1MAPTALOX5F10F7
SCHEMBL12366096 0.81 L3MBTL1 (0.57) MAPTHPGDL3MBTL1
SCHEMBL11591975 0.80 GAA (0.59) MAPTLMNACYP2C19HPGDL3MBTL1
SCHEMBL17570500 0.80 AOC3 (0.65) NPC1MAPTALOX5F10F7
SCHEMBL4075832 0.80 GAA (0.64) NPC1MAPTALOX5MTORLMNA
SCHEMBL30259901 0.80 NPC1 (0.59) NPC1MAPTALOX5F10F7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998986-B2 Heterocyclic compounds, in particular N-substituted pyridones for modulating the activity of nuclear receptors EXELIXIS PATENT COMPANY LLC (US) 2011-08-16 US disclosed