SCHEMBL12366208

SCHEMBL12366208

[C-]#[N+]CC(=O)NCc1cccc(F)c1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SRC P12931 2/20 0.57
RAB9A P51151 2/20 0.56
MAPK1 P28482 1/20 0.56
POLB P06746 2/20 0.53
TP53 P04637 1/20 0.51
ALDH1A1 P00352 1/20 0.49
KMT2A Q03164 1/20 0.47
KDM4E B2RXH2 1/20 0.47
HSD17B10 Q99714 1/20 0.47
FOLH1 Q04609 1/20 0.46
CHRM2 P08172 1/20 0.46
CHRM4 P08173 1/20 0.46
CHRM1 P11229 1/20 0.46
CHRM3 P20309 1/20 0.46
CNR1 P21554 1/20 0.46
ANPEP P15144 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18095012 0.83 SRC (0.61) SRCRAB9AMAPK1POLBTP53
SCHEMBL12366093 0.82 MMP13 (0.52) RAB9APOLBTP53ALDH1A1KDM4E
SCHEMBL12366183 0.82 NPC1 (0.56) TP53
SCHEMBL12366113 0.81 L3MBTL1 (0.63) RAB9APOLBALDH1A1KMT2A
SCHEMBL12366135 0.81 LMNA (0.62) RAB9APOLBTP53ALDH1A1KMT2A
SCHEMBL11591975 0.80 GAA (0.59) RAB9AALDH1A1KMT2A
SCHEMBL12366168 0.80 P2RX7 (0.44) ALDH1A1KMT2A
SCHEMBL5390715 0.80 SRC (0.61) SRCRAB9AMAPK1POLBTP53
SCHEMBL28822092 0.80 SRC (0.61) SRCRAB9AMAPK1POLBTP53
SCHEMBL4032122 0.80 ALDH1A1 (0.61) SRCRAB9AMAPK1POLBTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998986-B2 Heterocyclic compounds, in particular N-substituted pyridones for modulating the activity of nuclear receptors EXELIXIS PATENT COMPANY LLC (US) 2011-08-16 US disclosed