SCHEMBL12418540

SCHEMBL12418540

CCCCOc1ccc2c(c1)CCC1C2CC[C@]2(C)C(=O)C(CC(=O)O/N=C(\c3ccc(C)cc3)c3ccc([N+](=O)[O-])cc3)CC12

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 7/20 0.53
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
ZAP70 P43403 3/20 0.41
HRH3 Q9Y5N1 5/20 0.39
KCNH2 Q12809 3/20 0.39
FOLH1 Q04609 1/20 0.38
CYP3A4 P08684 1/20 0.38
CTRC Q99895 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12379546 0.91 HSD17B1 (0.51) HSD17B1KDM4EALDH1A1HRH3CYP3A4
SCHEMBL12379513 0.90 HSD17B1 (0.64) HSD17B1CYP3A4
SCHEMBL12418537 0.82 HSD17B1 (0.78) HSD17B1KDM4EALDH1A1ZAP70HRH3
SCHEMBL12418539 0.79 HSD17B1 (0.63) HSD17B1KDM4EALDH1A1CYP3A4
SCHEMBL12379510 0.72 HSD17B1 (0.76) HSD17B1KDM4EALDH1A1HRH3CYP3A4
SCHEMBL12379501 0.70 HSD17B1 (1.00) HSD17B1CYP3A4
SCHEMBL12379457 0.70 ESR1 (0.48) HSD17B1CYP3A4
SCHEMBL12418333 0.70 HSD17B1 (0.63) HSD17B1KDM4EALDH1A1HRH3CYP3A4
SCHEMBL7124873 0.69 HSD17B1 (0.64) HSD17B1KDM4EALDH1A1CYP3A4
SCHEMBL7124870 0.69 HSD17B1 (0.64) HSD17B1KDM4EALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8003783-B2 Steroid 17 beta -hydroxysteroid dehydrogenase inhibitors substituted with one or more oxime groups, especially aromatase inhibitors used in the treatment of endocrine-dependent tumors, especially breast cancer STERIX LIMITED (GB) 2011-08-23 US disclosed