SCHEMBL12428674

SCHEMBL12428674

CS(=O)(=O)N1CCN(c2ccc(N3CCCC3=O)cc2COc2ccc3c(c2)OCCn2c-3c(C3CCCCC3)c3ccc(C(=O)O)nc32)CC1

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.31
ADAM17 P78536 1/20 0.31
PDE7A Q13946 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL771502 0.99 ADAM17 (0.30) PIK3CAADAM17PDE7A
SCHEMBL12428670 0.92 FFAR4 (0.34) PIK3CAADAM17
Hydrochloric Acid SCHEMBL772629 0.91 FFAR4 (0.34) PIK3CA
SCHEMBL10283203 0.89 PRKCA (0.38)
Hydrochloric Acid SCHEMBL772348 0.88 PRKCA (0.38)
SCHEMBL13476323 0.84
SCHEMBL12428671 0.82 TRPM8 (0.34)
Hydrochloric Acid SCHEMBL771301 0.82 TRPM8 (0.34)
SCHEMBL3785533 0.81 PRKCA (0.39)
SCHEMBL804172 0.80 PRKCA (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7977331-B1 Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2011-07-12 US disclosed
US-7977331-B1 Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2011-07-12 US disclosed