SCHEMBL12434372

SCHEMBL12434372

Cn1c(=O)n(CC2CCCCC2)c2ccccc21

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARG Q86W56 4/20 0.54
ALDH1A1 P00352 4/20 0.52
KDM4E B2RXH2 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
HSD17B10 Q99714 1/20 0.52
OPRM1 P35372 1/20 0.52
OPRK1 P41145 1/20 0.52
OPRL1 P41146 1/20 0.52
CYP1A2 P05177 1/20 0.50
HPGD P15428 1/20 0.49
CRHR1 P34998 2/20 0.47
CRHR2 Q13324 1/20 0.47
TSHR P16473 2/20 0.47
NPC1 O15118 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2680469 0.92 CYP1A2 (0.54) PARGALDH1A1CYP1A2CRHR1CRHR2
SCHEMBL25720574 0.85 CYP1A2 (0.48) PARGALDH1A1CYP1A2CRHR1CRHR2
SCHEMBL12434220 0.84 OPRL1 (0.66) PARGALDH1A1KDM4ENPSR1HSD17B10
Hydrochloric Acid SCHEMBL2264513 0.84 CRHR1 (0.47) PARGALDH1A1CYP1A2CRHR1CRHR2
SCHEMBL11247925 0.83 BRD4 (0.52) PARGCYP1A2KMT2A
SCHEMBL12434209 0.80 CRHR1 (0.52) PARGALDH1A1KDM4ENPSR1HSD17B10
SCHEMBL12434217 0.80 ALDH1A1 (0.49) PARGALDH1A1KDM4ENPSR1HSD17B10
SCHEMBL24405966 0.80 OPRL1 (0.68) ALDH1A1KDM4ENPSR1HSD17B10OPRM1
SCHEMBL11949817 0.78 CRHR1 (0.51) ALDH1A1HSD17B10HPGDCRHR1CRHR2
SCHEMBL2149287 0.77 OPRM1 (0.46) OPRM1OPRK1OPRL1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011092293-A2 CYCLOHEXYL AMIDE DERIVATIVES AS CRF RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2011-08-04 WO disclosed