SCHEMBL12439665

SCHEMBL12439665

COc1cc(C(F)(F)F)cc(C2CC2)c1C(N)=O

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 1/20 0.42
HTR2A P28223 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.39
MRGPRX4 Q96LA9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL422861 0.87 MRGPRX4 (0.43) SLC9A1HTR2APTGDR2MRGPRX4
SCHEMBL30995068 0.78 HTR2A (0.44) SLC9A1HTR2APTGDR2
SCHEMBL26487993 0.78 MAP2K1 (0.41)
SCHEMBL25085869 0.75 HTR2A (0.44) SLC9A1HTR2APTGDR2MRGPRX4
SCHEMBL12439663 0.74 SLC6A9 (0.46)
SCHEMBL421430 0.73
SCHEMBL10189611 0.73
SCHEMBL421721 0.72 CA12 (0.52)
SCHEMBL6908816 0.71 IDO1 (0.38) SLC9A1HTR2APTGDR2MRGPRX4
SCHEMBL423901 0.71 GPR35 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011095434-A1 TETRAHYDRO-PYRAN DERIVATIVES AGAINST NEUROLOGICAL ILLNESSES F. HOFFMANN-LA ROCHE AG (CH) 2011-08-11 WO disclosed