SCHEMBL26487993

SCHEMBL26487993

COc1cc(C(F)(F)F)cc(F)c1C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 1/20 0.41
TGFBR1 P36897 4/20 0.38
ACVR1 Q04771 4/20 0.38
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
KDM4E B2RXH2 2/20 0.37
POLB P06746 1/20 0.37
CTDSP1 Q9GZU7 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GPBAR1 Q8TDU6 2/20 0.36
NOTUM Q6P988 1/20 0.36
BMPR1B O00238 1/20 0.36
BMPR1A P36894 1/20 0.36
ACVR1B P36896 1/20 0.36
ACVRL1 P37023 1/20 0.36
TNIK Q9UKE5 1/20 0.36
KCNH2 Q12809 1/20 0.36
MAPT P10636 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31092882 0.85 LMNA (0.44) AKR1C3AKR1C2KDM4ENOTUMUSP2
SCHEMBL26488238 0.85 LMNA (0.44) AKR1C3AKR1C2KDM4ENOTUMUSP2
SCHEMBL22093638 0.82 CES2 (0.45) KDM4EMAPTKMT2ALMNA
SCHEMBL12439663 0.80 SLC6A9 (0.46)
SCHEMBL12439665 0.78 SLC9A1 (0.42)
SCHEMBL421721 0.78 CA12 (0.52) AKR1C3AKR1C2KDM4ENOTUMUSP2
SCHEMBL22093825 0.77 DGAT1 (0.43) MAP2K1TGFBR1ACVR1KDM4EPOLB
SCHEMBL26486063 0.77 MAP2K1 (0.43) MAP2K1TGFBR1ACVR1KDM4EPOLB
SCHEMBL423901 0.76 GPR35 (0.41) AKR1C3AKR1C2KDM4ENOTUMMAPT
SCHEMBL14817465 0.76 NOTUM (0.51) AKR1C3AKR1C2KDM4ENOTUMMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024217493-A1 CRYSTALLINE METHIONINE ADENOSYLTRANSFERASE 2a (MAT2A) INHIBITOR AND USES THEREOF INSILICO MEDICINE IP LIMITED (CN) 2024-10-24 WO disclosed
WO-2023066283-A1 METHIONINE ADENOSYLTRANSFERASE 2A (MAT2A) INHIBITORS AND USES THEREOF INSILICO MEDICINE IP LIMITED (CN) 2023-04-27 WO disclosed