SCHEMBL6908816

SCHEMBL6908816

CC(=O)c1c(C2CC2)cc(C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.38
RBP4 P02753 2/20 0.37
CES2 O00748 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.36
SLC9A1 P19634 3/20 0.35
MRGPRX4 Q96LA9 1/20 0.35
ADRA1D P25100 1/20 0.35
HTR2A P28223 1/20 0.35
SLC6A3 Q01959 1/20 0.35
SLC9A2 Q9UBY0 1/20 0.35
CACNA1H O95180 1/20 0.35
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL422975 0.86 MRGPRX4 (0.41) RBP4CES2PTGDR2MRGPRX4
SCHEMBL30628783 0.81 CES2 (0.47) CES2CACNA1H
SCHEMBL6910600 0.75 KIF11 (0.42) CES2
SCHEMBL16449430 0.73 PTGDR2 (0.46) CES2PTGDR2
SCHEMBL16398462 0.73 MRGPRX4 (0.41) IDO1CES2PTGDR2MRGPRX4
SCHEMBL6909178 0.72 CES2 (0.40) CES2CACNA1H
SCHEMBL16398013 0.72 PTGDR2 (0.36) IDO1CES2PTGDR2MRGPRX4
SCHEMBL422861 0.72 MRGPRX4 (0.43) PTGDR2SLC9A1MRGPRX4HTR2A
SCHEMBL422141 0.71 RBP4 (0.33) IDO1RBP4CES2PTGDR2MRGPRX4
SCHEMBL12439665 0.71 SLC9A1 (0.42) PTGDR2SLC9A1MRGPRX4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011023667-A1 CARBOCYCLIC GLYT1 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2011-03-03 WO disclosed