SCHEMBL12445479

SCHEMBL12445479

CNC(=O)CCc1cccc(NC(=O)c2cnc(OCC3CCO3)cn2)c1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 15/20 0.58
PARP1 P09874 1/20 0.41
GRM4 Q14833 2/20 0.40
BACE2 Q9Y5Z0 1/20 0.40
ACKR3 P25106 1/20 0.40
GRM5 P41594 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12445770 0.82 BACE1 (0.51) BACE1BACE2
SCHEMBL12445476 0.82 BACE1 (0.61) BACE1
SCHEMBL12446184 0.82 BACE1 (0.53) BACE1PARP1
SCHEMBL12446154 0.81 BACE1 (0.54) BACE1PARP1
SCHEMBL12445462 0.80 BACE1 (0.55) BACE1PARP1
SCHEMBL7933976 0.77 BACE1 (0.72) BACE1GRM4BACE2
SCHEMBL7942075 0.77 ALDH1A1 (0.51) BACE1PARP1
SCHEMBL12445871 0.75 BACE1 (0.47) BACE1GRM4BACE2
SCHEMBL7943333 0.74 HDAC1 (0.48) BACE1
SCHEMBL4079617 0.73 BACE1 (1.00) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2360155-A1 2-AMINOPYRIDIN-4-ONE AND 2-AMINOPYRIDINE DERIVATIVE BOTH HAVING BACE1-INHIBITING ACTIVITY Shionogi & Co., Ltd. (JP) 2011-08-24 EP disclosed