SCHEMBL7943333

SCHEMBL7943333

CNC(=O)CCc1cccc(NC(=O)c2ccc(Br)cn2)c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.48
HDAC6 Q9UBN7 2/20 0.48
BACE1 P56817 7/20 0.46
APP P05067 3/20 0.46
ALDH1A1 P00352 3/20 0.44
MEN1 O00255 2/20 0.44
LMNA P02545 2/20 0.44
KMT2A Q03164 2/20 0.44
POLB P06746 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MAPT P10636 2/20 0.44
GAA P10253 1/20 0.44
ALOX15 P16050 1/20 0.43
ALOX12 P18054 1/20 0.43
SENP1 Q9P0U3 1/20 0.43
BRD4 O60885 1/20 0.42
TSHR P16473 1/20 0.42
CTSD P07339 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7942075 0.87 ALDH1A1 (0.51) HDAC1HDAC6BACE1ALDH1A1MEN1
SCHEMBL7941942 0.82 SORT1 (0.41) BACE1APPTSHR
SCHEMBL12446162 0.81 ALOX15 (0.47) HDAC1HDAC6ALDH1A1LMNAMAPT
SCHEMBL7942651 0.80 BACE1 (0.47) BACE1APPSMN1; SMN2
SCHEMBL12445826 0.80 SMN1; SMN2 (0.58) ALDH1A1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL12445476 0.79 BACE1 (0.61) BACE1
SCHEMBL12446184 0.79 BACE1 (0.53) HDAC1HDAC6BACE1
SCHEMBL12445770 0.79 BACE1 (0.51) BACE1
SCHEMBL12446169 0.78 BACE1 (0.47) HDAC1HDAC6BACE1ALDH1A1MEN1
SCHEMBL12446154 0.77 BACE1 (0.54) HDAC1HDAC6BACE1ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010047372-A1 2-AMINOPYRIDIN-4-ONE AND 2-AMINOPYRIDINE DERIVATIVE BOTH HAVING BACE1-INHIBITING ACTIVITY 塩野義製薬株式会社 (JP) 2010-04-29 WO disclosed