SCHEMBL12445826

SCHEMBL12445826

CNC(=O)CCc1cccc(NC(=O)c2cnc3ccccc3n2)c1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.58
RAB9A P51151 5/20 0.57
NPC1 O15118 4/20 0.57
MAPT P10636 3/20 0.57
MEN1 O00255 1/20 0.57
ALDH1A1 P00352 1/20 0.57
ABCB1 P08183 1/20 0.57
HTT P42858 1/20 0.57
KMT2A Q03164 1/20 0.57
ABCG2 Q9UNQ0 1/20 0.57
GAA P10253 1/20 0.57
ACKR3 P25106 1/20 0.53
RHOA P61586 1/20 0.53
KDM4E B2RXH2 1/20 0.49
CBLB Q13191 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7942075 0.81 ALDH1A1 (0.51) SMN1; SMN2RAB9ANPC1MAPTMEN1
SCHEMBL7943333 0.80 HDAC1 (0.48) SMN1; SMN2MAPTMEN1ALDH1A1KMT2A
SCHEMBL12446162 0.79 ALOX15 (0.47) RAB9AMAPTALDH1A1GAAACKR3
SCHEMBL12446184 0.77 BACE1 (0.53)
SCHEMBL12445770 0.77 BACE1 (0.51)
SCHEMBL12445476 0.77 BACE1 (0.61)
SCHEMBL12446169 0.76 BACE1 (0.47) SMN1; SMN2RAB9ANPC1MAPTMEN1
SCHEMBL12446154 0.76 BACE1 (0.54) ALDH1A1
SCHEMBL12445462 0.75 BACE1 (0.55)
SCHEMBL12445472 0.74 BACE1 (0.41) RAB9AMAPTALDH1A1GAAACKR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2360155-A1 2-AMINOPYRIDIN-4-ONE AND 2-AMINOPYRIDINE DERIVATIVE BOTH HAVING BACE1-INHIBITING ACTIVITY Shionogi & Co., Ltd. (JP) 2011-08-24 EP disclosed