SCHEMBL12445904

SCHEMBL12445904

C=C/C=C\C(NCc1cc(NC(=O)c2sc3ccc(O)cc3c2C)ccc1F)=C(N)N

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.38
F10 P00742 6/20 0.36
CISD2 Q8N5K1 4/20 0.33
CXCR2 P25025 1/20 0.33
ICAM1 P05362 1/20 0.32
SELE P16581 1/20 0.32
MAOB P27338 1/20 0.32
BRD4 O60885 1/20 0.31
SENP5 Q96HI0 1/20 0.31
SENP2 Q9HC62 1/20 0.31
SENP1 Q9P0U3 1/20 0.31
AURKA O14965 1/20 0.31
AURKB Q96GD4 1/20 0.31
LMNA P02545 2/20 0.30
NPC1 O15118 1/20 0.30
MAPT P10636 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12445797 0.85 F10 (0.34) PTGDR2F10CISD2CXCR2ICAM1
SCHEMBL7940504 0.73 PTGDR2 (0.40) PTGDR2F10CISD2CXCR2AURKA
SCHEMBL12446317 0.73 BACE1 (0.41) AURKAAURKBNPC1RAB9A
SCHEMBL12445900 0.67 BACE1 (0.42)
SCHEMBL7943357 0.62 BACE1 (0.52)
SCHEMBL7942773 0.60 BACE1 (0.41) F10CISD2
SCHEMBL7945236 0.60 BACE1 (0.54) SENP5SENP2SENP1MAPT
SCHEMBL9757077 0.59 GPR35 (0.65) ICAM1SELE
SCHEMBL9756981 0.58 MAPK1 (0.53) CISD2ICAM1SELELMNAMAPT
SCHEMBL20838905 0.58 ADORA1 (0.67) CISD2NPC1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2360155-A1 2-AMINOPYRIDIN-4-ONE AND 2-AMINOPYRIDINE DERIVATIVE BOTH HAVING BACE1-INHIBITING ACTIVITY Shionogi & Co., Ltd. (JP) 2011-08-24 EP disclosed