SCHEMBL9757077

SCHEMBL9757077

Cc1c(C(=O)O)sc2ccc(O)cc12

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 5/20 0.65
TBXAS1 P24557 3/20 0.50
RXFP1 Q9HBX9 3/20 0.49
PKM P14618 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
ICAM1 P05362 1/20 0.48
SELE P16581 1/20 0.48
PRNP P04156 1/20 0.45
MCL1 Q07820 4/20 0.44
BCL2L1 Q07817 2/20 0.44
CLK1 P49759 1/20 0.40
DYRK1A Q13627 1/20 0.40
DYRK1B Q9Y463 1/20 0.40
CA12 O43570 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
TSHR P16473 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2895952 0.84 GPR35 (0.62) GPR35TBXAS1RXFP1PKMNPSR1
SCHEMBL9756981 0.82 MAPK1 (0.53) GPR35PKMICAM1SELECA12
SCHEMBL2893771 0.81 GPR35 (0.58) GPR35TBXAS1RXFP1PKMNPSR1
SCHEMBL122587 0.81 GPR35 (0.58) GPR35TBXAS1RXFP1PKMNPSR1
SCHEMBL1066852 0.81 GPR35 (0.58) GPR35TBXAS1RXFP1PKMNPSR1
SCHEMBL2896475 0.81 GPR35 (0.58) GPR35TBXAS1RXFP1PKMNPSR1
SCHEMBL3484085 0.80 GPR35 (0.57) GPR35TBXAS1RXFP1PKMNPSR1
SCHEMBL14691616 0.80 CA12 (0.53) NPSR1ICAM1SELECA12ALDH1A1
SCHEMBL10948748 0.79 TBXAS1 (0.60) GPR35TBXAS1RXFP1PKMNPSR1
SCHEMBL9613211 0.79 TBXAS1 (0.60) GPR35TBXAS1RXFP1PKMNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019475-A2 QUINOLINYL-BENZOHETEROBICYCLIC DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D¿4? RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1991-12-26 WO disclosed
US-5041453-A Quinolinyl-benzoheterobicyclic derivatives as antagonists of leukotriene D4 RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-08-20 US disclosed