SCHEMBL1245262

SCHEMBL1245262

CCOC(=O)N(c1ccc(F)cc1F)c1c(-c2ccc(-c3ccc(CC(=O)O)cc3)cc2)noc1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.37
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 2/20 0.35
GAA P10253 2/20 0.35
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPC1 O15118 2/20 0.35
DGAT1 O75907 2/20 0.35
SOAT1 P35610 1/20 0.35
FFAR4 Q5NUL3 2/20 0.35
RXRA P19793 2/20 0.35
RXRB P28702 2/20 0.35
RXRG P48443 2/20 0.35
GABRA5 P31644 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ATM Q13315 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1247624 0.93 THRB (0.37) THRBALDH1A1KDM4EGAALMNA
SCHEMBL1246439 0.91 PPARD (0.37) ALDH1A1DGAT1SOAT1FFAR4MEN1
SCHEMBL1247343 0.90 PTGS2 (0.42) NPC1FFAR4RXRARXRBRXRG
SCHEMBL1245270 0.89 KDM4E (0.44) ALDH1A1KDM4EGAALMNAHPGD
SCHEMBL1247569 0.86 SCN9A (0.39) KDM4ENPC1DGAT1CACNA1FCACNA1D
SCHEMBL2337987 0.85 LPAR1 (0.40) DGAT1SOAT1RXRARXRBRXRG
SCHEMBL1247291 0.85 SCN9A (0.41) KDM4EGAALMNANPC1DGAT1
SCHEMBL1247301 0.84 PPARD (0.41) ALDH1A1MEN1KMT2A
SCHEMBL1246323 0.83 PPARD (0.39) ALDH1A1KDM4EGAALMNAHPGD
SCHEMBL1247349 0.83 GPBAR1 (0.39) ALDH1A1KDM4EGAALMNADGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2462128-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-06-13 EP claimed
WO-2011017350-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-02-10 WO claimed