SCHEMBL12461572

SCHEMBL12461572

Bc1ccc(-c2ncc(C)s2)nc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SRC P12931 2/20 0.39
ZAP70 P43403 2/20 0.39
SYK P43405 2/20 0.39
CDK2 P24941 1/20 0.39
NOS1 P29475 1/20 0.36
CCR1 P32246 1/20 0.34
CCR5 P51681 1/20 0.34
CCR8 P51685 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
ALDH1A1 P00352 1/20 0.32
HDAC4 P56524 1/20 0.31
SCD O00767 1/20 0.31
MET P08581 1/20 0.30
KDR P35968 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12460344 0.81 CCR1 (0.58) SRCZAP70SYKCDK2NOS1
SCHEMBL15633091 0.78 CYP2C9 (0.40) SRCZAP70SYKCDK2NOS1
SCHEMBL14298327 0.78 SRC (0.39) SRCZAP70SYKCDK2NOS1
SCHEMBL13676792 0.75
SCHEMBL20068615 0.72 CCR1 (0.46) CCR1CCR5CCR8HDAC6ALDH1A1
SCHEMBL10002194 0.72 NOS1 (0.55) SRCZAP70SYKCDK2NOS1
SCHEMBL12116515 0.72 ALDH1A1 (0.58) SRCZAP70SYKCDK2CCR1
SCHEMBL805859 0.70 RAB9A (0.60) ALDH1A1
SCHEMBL2147093 0.68 DGAT1 (0.45) SRCZAP70SYKCDK2KDR
SCHEMBL20175446 0.67 NOS1 (0.44) SRCZAP70SYKCDK2NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011090935-A1 PYRAZOLO[1,5-a]PYRIMIDINE COMPOUNDS AS mTOR INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-07-28 WO disclosed