SCHEMBL1246320

SCHEMBL1246320

CCOC(=O)N(c1ccccc1F)c1c(-c2ccc(-c3ccc(C(C)(C)C(=O)O)cc3)cc2)noc1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.39
CACNA1F O60840 1/20 0.39
CACNA1D Q01668 1/20 0.39
CACNA1S Q13698 1/20 0.39
CACNA1C Q13936 1/20 0.39
KDM4E B2RXH2 3/20 0.38
PPARG P37231 1/20 0.38
PPARD Q03181 1/20 0.38
PPARA Q07869 1/20 0.38
SCN9A Q15858 1/20 0.37
MAPT P10636 1/20 0.36
GPBAR1 Q8TDU6 1/20 0.36
NR1H4 Q96RI1 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MLYCD O95822 2/20 0.36
TSHR P16473 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1247617 0.91 NPC1 (0.38) NPC1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL1245152 0.90 NR1H4 (0.42) CACNA1FCACNA1DCACNA1SCACNA1CKDM4E
SCHEMBL1245270 0.86 KDM4E (0.44) NPC1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL2338970 0.85 USP2 (0.35) KDM4EPPARGPPARDPPARAMAPT
SCHEMBL1246242 0.84 PTGS2 (0.39) NPC1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL1247569 0.80 SCN9A (0.39) NPC1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL2335133 0.78 TP53 (0.34) KDM4EMAPTALDH1A1MLYCDTSHR
SCHEMBL1247556 0.78 KDM4E (0.40) NPC1KDM4EPPARGPPARDPPARA
SCHEMBL1246914 0.77 KDM4E (0.39) NPC1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL1247289 0.77 KDM4E (0.39) NPC1CACNA1FCACNA1DCACNA1SCACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2462128-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-06-13 EP claimed
WO-2011017350-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-02-10 WO claimed