SCHEMBL1245152

SCHEMBL1245152

CCOC(=O)N(c1ccccc1Cl)c1c(-c2ccc(-c3ccc(C(C)(C)C(=O)O)cc3)cc2)noc1C

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.42
GPBAR1 Q8TDU6 7/20 0.38
MAPT P10636 2/20 0.38
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
HPGD P15428 1/20 0.38
PPARG P37231 1/20 0.37
PPARD Q03181 1/20 0.37
PPARA Q07869 1/20 0.37
FABP1 P07148 1/20 0.37
SCN9A Q15858 1/20 0.37
PTGS2 P35354 1/20 0.37
CACNA1F O60840 1/20 0.36
CACNA1D Q01668 1/20 0.36
CACNA1S Q13698 1/20 0.36
CACNA1C Q13936 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1246320 0.90 NPC1 (0.39) NR1H4GPBAR1MAPTALDH1A1POLB
SCHEMBL1247564 0.87 MAPT (0.42) NR1H4GPBAR1MAPTALDH1A1POLB
SCHEMBL2338001 0.85 NR1H4 (0.39) NR1H4MAPTALDH1A1HPGDPPARG
SCHEMBL1245358 0.85 NR1H4 (0.42) NR1H4GPBAR1MAPTALDH1A1POLB
SCHEMBL1245116 0.84 PTGS2 (0.39) GPBAR1MAPTALDH1A1POLBHPGD
SCHEMBL1247211 0.84 FFAR4 (0.42) NR1H4GPBAR1MAPTALDH1A1POLB
SCHEMBL1245320 0.83 NR1H4 (0.45) NR1H4GPBAR1MAPTALDH1A1POLB
SCHEMBL1246504 0.83 GPBAR1 (0.38) GPBAR1MAPTALDH1A1POLBHPGD
SCHEMBL1245150 0.83 GPBAR1 (0.39) GPBAR1MAPTALDH1A1POLBHPGD
SCHEMBL1247806 0.83 GPBAR1 (0.43) NR1H4GPBAR1MAPTALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2462128-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-06-13 EP claimed
WO-2011017350-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-02-10 WO claimed