SCHEMBL1247556

SCHEMBL1247556

CCOC(=O)N(c1ccccc1F)c1c(-c2ccc(Oc3cccc(CC(=O)O)c3)cc2)noc1C

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
PPARG P37231 2/20 0.38
PPARD Q03181 2/20 0.38
PPARA Q07869 2/20 0.38
NR3C1 P04150 3/20 0.38
SRD5A2 P31213 2/20 0.37
PTGDR2 Q9Y5Y4 3/20 0.36
TP53 P04637 1/20 0.36
FFAR1 O14842 1/20 0.36
SCN9A Q15858 2/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1247798 0.92 KDM4E (0.37) KDM4ETP53SCN9ANPC1
SCHEMBL1245136 0.90 NR1H4 (0.38) PPARGPPARDPPARANR3C1PTGDR2
SCHEMBL1245270 0.87 KDM4E (0.44) KDM4EPPARDTP53SCN9ANPC1
SCHEMBL3712290 0.87 NR3C1 (0.38) KDM4ENR3C1SRD5A2PTGDR2TP53
SCHEMBL1247289 0.86 KDM4E (0.39) KDM4EPPARGPPARDPPARATP53
SCHEMBL1247569 0.83 SCN9A (0.39) KDM4EPPARDTP53SCN9ANPC1
SCHEMBL1246477 0.82 NR1H4 (0.42) PPARGPPARDPPARAPTGDR2
SCHEMBL1246914 0.80 KDM4E (0.39) KDM4EPPARGPPARDPPARATP53
SCHEMBL9902690 0.80 L3MBTL1 (0.42) KDM4EPPARGSCN9ANPC1
SCHEMBL1247343 0.80 PTGS2 (0.42) PPARDFFAR1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2462128-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-06-13 EP claimed
WO-2011017350-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-02-10 WO claimed