SCHEMBL12465708

SCHEMBL12465708

CCCC(CCc1cc(F)c2c(c1)C(C)(C)CCO2)C(C)=O

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SSTR5 P35346 4/20 0.40
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
RXRA P19793 3/20 0.31
RARA P10276 1/20 0.31
RARB P10826 1/20 0.31
RARG P13631 1/20 0.31
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31
RXRB P28702 1/20 0.30
RXRG P48443 1/20 0.30
HNF4A P41235 2/20 0.30
CYP26A1 O43174 1/20 0.30
CYP26B1 Q9NR63 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12465704 0.81 CYP26A1 (0.45) SSTR5RXRARARARARBRARG
SCHEMBL12468551 0.68 PTGS2 (0.40) SSTR5PTGS1PTGS2RXRARARA
SCHEMBL12465698 0.66 PTGS2 (0.46) SSTR5PTGS1PTGS2RXRARARA
SCHEMBL12465974 0.65 NOTUM (0.33)
SCHEMBL12465596 0.63 MME (0.41) TAS1R3TAS1R1
SCHEMBL12465699 0.61 SSTR5 (0.33) SSTR5PTGS1PTGS2
SCHEMBL15002369 0.61 PTGS1 (0.35) SSTR5PTGS1PTGS2RXRAHNF4A
SCHEMBL7196161 0.60 SSTR5 (0.38) SSTR5PTGS1PTGS2RXRARARA
SCHEMBL9766489 0.60 HDAC1 (0.60)
SCHEMBL12465678 0.59 SSTR5 (0.33) SSTR5RARARARBRARGHNF4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2670744-A1 PYRROLE DERIVATIVES USED AS MODULATORS OF ALPHA7 NACHR Lupin Limited (IN) 2013-12-11 EP disclosed
WO-2012104782-A1 PYRROLE DERIVATIVES USED AS MODULATORS OF ALPHA7 NACHR LUPIN LIMITED (IN) 2012-08-09 WO disclosed