SCHEMBL7196161

SCHEMBL7196161

CC1(C)CCOc2c(N)cc(CC(=O)Cc3cc(N)c4c(c3)C(C)(C)CCO4)cc21

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SSTR5 P35346 6/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
CYP26A1 O43174 4/20 0.37
CYP26B1 Q9NR63 3/20 0.37
HNF4A P41235 2/20 0.35
RARA P10276 4/20 0.34
RARB P10826 4/20 0.34
RARG P13631 4/20 0.34
RXRA P19793 4/20 0.33
RXRB P28702 2/20 0.33
RXRG P48443 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7196167 0.81 PTGS1 (0.34) SSTR5PTGS1PTGS2CYP26A1CYP26B1
SCHEMBL7183938 0.79 HNF4A (0.44) SSTR5PTGS1PTGS2CYP26A1CYP26B1
SCHEMBL7196169 0.77 PTGS1 (0.42) SSTR5PTGS1PTGS2CYP26A1CYP26B1
SCHEMBL11241526 0.67 RXRA (0.60) CYP26A1CYP26B1RARARARBRARG
SCHEMBL6146899 0.66 CYP26A1 (0.69) SSTR5CYP26A1CYP26B1HNF4ARARA
SCHEMBL2053058 0.65 CYP26A1 (0.46) SSTR5CYP26A1CYP26B1HNF4ARARA
SCHEMBL12182489 0.64 PTGS1 (0.41) SSTR5PTGS1PTGS2CYP26A1CYP26B1
SCHEMBL15002369 0.63 PTGS1 (0.35) SSTR5PTGS1PTGS2CYP26A1CYP26B1
SCHEMBL3584479 0.62 PTGS2 (0.62) PTGS1PTGS2
SCHEMBL21911671 0.62 PARP1 (0.54) HNF4ARARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6586460-B1 Administering heterocyclic ethers or sulfides to induce apoptosis, cell differentiation and as anticarcinogenic agents THE BOARD OF REGENTS FOR OKLAHOMA STATE UNIVERSITY 2003-07-01 US disclosed