SCHEMBL12466762

SCHEMBL12466762

Cc1cccc(CON=CCc2ccc(Cl)c(CNC(=O)O)c2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.38
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
MAOB P27338 2/20 0.37
OPRK1 P41145 1/20 0.36
HSP90AA1 P07900 1/20 0.36
CTBP2 P56545 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.36
IDO1 P14902 2/20 0.36
THRA P10827 1/20 0.35
THRB P10828 1/20 0.35
FFAR4 Q5NUL3 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
MAPT P10636 2/20 0.35
MAPK1 P28482 1/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
CXCR4 P61073 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17845833 0.93 TSHR (0.42) PPARGKMT2AMEN1MAOBOPRK1
SCHEMBL166893 0.85 KDM4E (0.41) KMT2AMEN1MAOBHSP90AA1CTBP2
SCHEMBL9958047 0.84 IDO1 (0.39) KMT2AMEN1MAOBHSP90AA1CTBP2
SCHEMBL9954743 0.83 PTGES (0.39) KMT2AMEN1OPRK1MRGPRX4L3MBTL1
SCHEMBL26317 0.78 NPC1 (0.53) PPARGKMT2AMEN1MAOBHSP90AA1
SCHEMBL26318 0.78 NPC1 (0.53) PPARGKMT2AMEN1MAOBHSP90AA1
SCHEMBL2781697 0.78 IDO1 (0.42) KMT2AMEN1MAOBHSP90AA1IDO1
SCHEMBL482900 0.77 TSHR (0.40) KMT2AMEN1MRGPRX4MAPT
SCHEMBL1274673 0.75 IDO1 (0.36) KMT2AMEN1MAOBHSP90AA1MRGPRX4
SCHEMBL4667807 0.73 NPC1 (0.48) PPARGKMT2AMEN1MAOBHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 48 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020206518-A1 MULTIPURPOSE BIOLOGICAL COMPOSITIONS AGRIVALLE BRASIL INDUSTRIA E COMÉRCIO DE PRODUTOS AGRÍCOLAS LTDA (BR) 2020-10-15 WO claimed
EP-3634130-A1 COMBINATION OF PYROGLUTAMIC ACID AND A STROBILURIN FUNGICIDE FOR IMPROVED PLANT HEALTH EFFECTS Verdesian Life Sciences U.S., LLC (US) 2020-04-15 EP claimed
WO-2018224966-A1 COMBINATION OF PYROGLUTAMIC ACID AND A STROBILURIN FUNGICIDE FOR IMPROVED PLANT HEALTH EFFECTS VERDESIAN LIFE SCIENCES U.S., LLC (US) 2018-12-13 WO claimed
EP-3240406-A1 BACILLUS AMYLOLIQUEFACIENS RTI472 COMPOSITIONS AND METHODS OF USE FOR BENEFITING PLANT GROWTH AND TREATING PLANT DISEASE FMC CORPORATION (US) 2017-11-08 EP claimed
WO-2016109332-A1 COMPOSITIONS AND METHODS FOR USE OF INSECTICIDE WITH BACILLUS SP. D747 FMC CORPORATION (US) 2016-07-07 WO claimed
WO-2016109396-A1 BACILLUS AMYLOLIQUEFACIENS RTI472 COMPOSITIONS AND METHODS OF USE FOR BENEFITING PLANT GROWTH AND TREATING PLANT DISEASE FMC CORPORATION (US) 2016-07-07 WO claimed
WO-2022011298-A1 MICROALGAE AND FERTILIZER MIXTURES AND METHODS OF USE THEREOF TO ENHANCE PLANT CHARACTERISTICS HELIAE DEVELOPMENT LLC (US) 2022-01-13 WO disclosed
EP-3855919-A1 BACILLUS AMYLOLIQUEFACIENS FCC1256 COMPOSITIONS AND METHODS OF CONTROLLING PLANT PATHOGENS
 FMC Corporation (US) 2021-08-04 EP disclosed
WO-2020206518-A1 MULTIPURPOSE BIOLOGICAL COMPOSITIONS AGRIVALLE BRASIL INDUSTRIA E COMÉRCIO DE PRODUTOS AGRÍCOLAS LTDA (BR) 2020-10-15 WO disclosed
EP-3634130-A1 COMBINATION OF PYROGLUTAMIC ACID AND A STROBILURIN FUNGICIDE FOR IMPROVED PLANT HEALTH EFFECTS Verdesian Life Sciences U.S., LLC (US) 2020-04-15 EP disclosed
WO-2020069297-A1 BACILLUS AMYLOLIQUEFACIENS FCC1256 COMPOSITIONS AND METHODS OF CONTROLLING PLANT PATHOGENS FMC CORPORATION (US) 2020-04-02 WO disclosed
EP-3522706-A1 BACILLUS THURINGIENSIS FMC Corporation (US) 2019-08-14 EP disclosed
WO-2018224966-A1 COMBINATION OF PYROGLUTAMIC ACID AND A STROBILURIN FUNGICIDE FOR IMPROVED PLANT HEALTH EFFECTS VERDESIAN LIFE SCIENCES U.S., LLC (US) 2018-12-13 WO disclosed
WO-2015050918-A1 CO-FORMULATIONS OF BIFENTHRIN WITH ENCAPSULATED CROP PROTECTION AGENTS FOR USE WITH LIQUID FERTILIZERS FMC CORPORATION (US) 2015-04-09 WO disclosed
WO-2014182951-A1 ACC INHIBITORS AND USES THEREOF Nimbus Apollo, Inc. (US) 2014-11-13 WO disclosed
WO-2014177475-A1 CROP ENHANCEMENT SYNGENTA PARTICIPATIONS AG (CH) 2014-11-06 WO disclosed
EP-2776038-A1 ACC INHIBITORS AND USES THEREOF Nimbus Apollo Inc. (US) 2014-09-17 EP disclosed
EP-2611292-A1 NEONICOTINYL FORMULATIONS Cheminova A/S (DK) 2013-07-10 EP disclosed
WO-2013071169-A1 ACC INHIBITORS AND USES THEREOF Nimbus Apollo, Inc. (US) 2013-05-16 WO disclosed
WO-2012028151-A1 NEONICOTINYL FORMULATIONS CHEMINOVA A/S (DK) 2012-03-08 WO disclosed