SCHEMBL12469629

SCHEMBL12469629

NC(=O)c1ccc(-c2ccc(N)c(F)c2)c2c1C(=O)NC2.Nc1ccc(F)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.41
AURKA O14965 1/20 0.38
GRM2 Q14416 1/20 0.37
BTK Q06187 6/20 0.36
IKBKB O14920 3/20 0.35
CHUK O15111 3/20 0.35
PDE3B Q13370 2/20 0.34
PDE3A Q14432 2/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
CDC7 O00311 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12469765 0.85 AURKA (0.40) KDRAURKAGRM2BTKIKBKB
SCHEMBL18170475 0.75 KDR (0.52) KDRGRM2PDE3BPDE3APIK3CD
SCHEMBL1292744 0.75 AURKA (0.48) KDRAURKAPIK3CDPIK3CAPIK3CB
SCHEMBL12469562 0.73 BTK (0.42) KDRGRM2BTKIKBKBALOX5AP
SCHEMBL1292654 0.73 BTK (0.57) KDRAURKABTK
SCHEMBL12469505 0.71 BTK (0.41) KDRBTK
SCHEMBL29996262 0.71 IKBKB (0.46) IKBKBCHUKALOX5APFEN1CYP1A2
SCHEMBL1335395 0.71 PIK3CD (0.56) KDRAURKAGRM2PIK3CDPIK3CA
SCHEMBL12469512 0.71 CRBN (0.41) BTKALOX5APFEN1
SCHEMBL12469481 0.71 ALOX5 (0.40) KDRBTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047017-A2 2,3-DIHYDRO-ISOINDOL-1-ONE DERIVATIVE AND A COMPOSITION COMPRISING THE SAME 크리스탈지노믹스(주) (KR) 2012-04-12 WO disclosed