SCHEMBL12487524

SCHEMBL12487524

FC(F)(F)c1n[c]nc2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DCTPP1 Q9H773 1/20 0.41
KDM4E B2RXH2 3/20 0.38
MAPT P10636 2/20 0.38
BACE1 P56817 1/20 0.37
GAA P10253 3/20 0.36
ALDH1A1 P00352 3/20 0.36
ELANE P08246 1/20 0.36
PKM P14618 1/20 0.36
KHK P50053 1/20 0.36
GPR3 P46089 1/20 0.34
RAB9A P51151 1/20 0.34
CCNE2 O96020 2/20 0.33
CDK4 P11802 2/20 0.33
CCND1 P24385 2/20 0.33
CCNE1 P24864 2/20 0.33
CDK2 P24941 2/20 0.33
HPGD P15428 1/20 0.33
ENPP3 O14638 1/20 0.33
ENPP1 P22413 1/20 0.33
TLR7 Q9NYK1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2303106 0.80 ATM (0.36) KDM4EMAPTGAAALDH1A1ELANE
SCHEMBL28057497 0.69 GAA (0.61) DCTPP1MAPTGAAALDH1A1RAB9A
SCHEMBL7039137 0.68 GPR3 (0.39) KDM4EMAPTGAAALDH1A1GPR3
SCHEMBL637547 0.68 ALDH1A1 (0.45) KDM4EMAPTBACE1ALDH1A1ELANE
SCHEMBL558169 0.68 CYP1A2 (0.39) KDM4EMAPTGAAALDH1A1GPR3
SCHEMBL623055 0.68 DCPS (0.48) KDM4EMAPTGAAALDH1A1PKM
SCHEMBL7972478 0.68 PDE4A (0.48) KDM4EMAPTALDH1A1PKMGPR3
SCHEMBL28199808 0.67 GAA (0.50) DCTPP1KDM4EMAPTBACE1GAA
SCHEMBL20526115 0.67 BACE1 (0.51) KDM4EMAPTBACE1GAAALDH1A1
SCHEMBL30945013 0.67 DCPS (0.57) DCTPP1KDM4EMAPTBACE1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611502-A1 ADENOSINE A3 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF Ambit Biosciences Corporation (US) 2013-07-10 EP disclosed
WO-2012030918-A1 ADENOSINE A3 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2012-03-08 WO disclosed