SCHEMBL12499501

SCHEMBL12499501

C[C@@H]1CN(c2ccc(I)cc2)C[C@H](C)N1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 2/20 0.45
CCND1 P24385 2/20 0.45
TGFBR1 P36897 1/20 0.40
ACVR1 Q04771 1/20 0.40
KCNH2 Q12809 1/20 0.40
LTA4H P09960 1/20 0.40
GHSR Q92847 13/20 0.38
HTT P42858 1/20 0.36
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
AKR1C3 P42330 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL81349 0.82 ADRB1 (0.48) TGFBR1ACVR1KCNH2GHSRHTT
SCHEMBL81695 0.82 ADRB1 (0.48) TGFBR1ACVR1KCNH2GHSRHTT
SCHEMBL18711251 0.80 SIGMAR1 (0.46) TGFBR1ACVR1KCNH2GHSRHTT
SCHEMBL16069835 0.80 MAPT (0.47) TGFBR1ACVR1KCNH2GHSRHTT
SCHEMBL2446299 0.80 MAPT (0.47) TGFBR1ACVR1KCNH2GHSRHTT
SCHEMBL3528425 0.80 MAPT (0.47) TGFBR1ACVR1KCNH2GHSRHTT
SCHEMBL6367230 0.80 HTR3E (0.47) TGFBR1ACVR1KCNH2LTA4HGHSR
SCHEMBL2549111 0.80 GHSR (0.53) CDK4CCND1TGFBR1ACVR1KCNH2
SCHEMBL578246 0.80 GHSR (0.53) CDK4CCND1TGFBR1ACVR1KCNH2
SCHEMBL6367231 0.80 HTR3E (0.47) TGFBR1ACVR1KCNH2LTA4HGHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012048411-A1 PLK-4 INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2012-04-19 WO disclosed