SCHEMBL12503222

SCHEMBL12503222

Clc1ccc(C(c2nnn[nH]2)N2CCCCC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.47
CYP19A1 P11511 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.43
CHRM2 P08172 2/20 0.43
HTR1A P08908 2/20 0.43
ADRA2A P08913 2/20 0.43
CHRM1 P11229 2/20 0.43
DRD1 P21728 2/20 0.43
TBXA2R P21731 2/20 0.43
SLC6A2 P23975 2/20 0.43
SLC6A4 P31645 2/20 0.43
ADRA1A P35348 2/20 0.43
DRD3 P35462 2/20 0.43
SLC6A3 Q01959 2/20 0.43
KCNH2 Q12809 2/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP3A4 P08684 2/20 0.43
USP2 O75604 2/20 0.43
OPRM1 P35372 1/20 0.43
KDM4E B2RXH2 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL324172 0.87 CYP2D6 (0.67) CYP2D6CYP19A1CHRM2HTR1AADRA2A
SCHEMBL325002 0.86 ALDH1A1 (0.47) CYP2D6CYP19A1SMN1; SMN2CHRM2HTR1A
SCHEMBL323778 0.86 CHRM2 (0.58) CYP2D6CYP19A1SMN1; SMN2CHRM2HTR1A
SCHEMBL324760 0.85 ALDH1A1 (0.45) SMN1; SMN2SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL327686 0.83 CYP2D6 (0.43) CYP2D6CYP19A1SMN1; SMN2CHRM2HTR1A
SCHEMBL323776 0.80 CYP3A4 (0.61) CYP2D6CYP19A1CHRM2HTR1AADRA2A
SCHEMBL325153 0.79 CYP3A4 (0.48) CYP2D6CYP19A1CHRM2HTR1AADRA2A
SCHEMBL16757326 0.79 CYP2D6 (0.66) CYP2D6CYP19A1SMN1; SMN2CHRM2HTR1A
SCHEMBL323141 0.78 SLC6A9 (0.38) CYP2D6CYP19A1SLC6A2SLC6A4SLC6A3
SCHEMBL324763 0.76 CYP3A4 (0.45) CYP2D6CYP19A1CHRM2HTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2590953-A1 TETRAZOLE COMPOUNDS AS CALCIUM CHANNEL BLOCKERS Convergence Pharmaceuticals Limited (GB) 2013-05-15 EP claimed
WO-2012004604-A1 TETRAZOLE COMPOUNDS AS CALCIUM CHANNEL BLOCKERS Convergence Pharmaceuticals Limited (GB) 2012-01-12 WO claimed