SCHEMBL324760

SCHEMBL324760

Clc1ccc(C(c2nnn[nH]2)N2CCCCC2)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
GAA P10253 1/20 0.45
ADAM17 P78536 1/20 0.45
MCL1 Q07820 1/20 0.45
SLC6A3 Q01959 9/20 0.43
SLC6A2 P23975 8/20 0.43
SLC6A4 P31645 7/20 0.43
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
HPGD P15428 1/20 0.35
POLB P06746 2/20 0.34
HTT P42858 2/20 0.34
HRH3 Q9Y5N1 1/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
HSP90AA1 P07900 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL325375 0.87 SLC6A2 (0.45) ALDH1A1MEN1KMT2ASMN1; SMN2GAA
SCHEMBL12503222 0.85 CYP2D6 (0.47) ALDH1A1MEN1KMT2ASMN1; SMN2SLC6A3
SCHEMBL324172 0.72 CYP2D6 (0.67) MEN1KMT2ASLC6A3SLC6A2SLC6A4
SCHEMBL323778 0.71 CHRM2 (0.58) ALDH1A1MEN1KMT2ASMN1; SMN2GAA
SCHEMBL325002 0.71 ALDH1A1 (0.47) ALDH1A1MEN1KMT2ASMN1; SMN2SLC6A3
SCHEMBL327686 0.69 CYP2D6 (0.43) ALDH1A1MEN1KMT2ASMN1; SMN2SLC6A3
SCHEMBL29585835 0.68 SLC6A3 (0.56) ALDH1A1MEN1KMT2ASMN1; SMN2GAA
SCHEMBL29585404 0.68 SLC6A3 (0.56) ALDH1A1MEN1KMT2ASMN1; SMN2GAA
SCHEMBL22206745 0.68 SLC6A3 (0.56) ALDH1A1MEN1KMT2ASMN1; SMN2GAA
SCHEMBL22206766 0.68 SLC6A3 (0.56) ALDH1A1MEN1KMT2ASMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2590953-A1 TETRAZOLE COMPOUNDS AS CALCIUM CHANNEL BLOCKERS Convergence Pharmaceuticals Limited (GB) 2013-05-15 EP claimed
WO-2012004604-A1 TETRAZOLE COMPOUNDS AS CALCIUM CHANNEL BLOCKERS Convergence Pharmaceuticals Limited (GB) 2012-01-12 WO claimed
EP-2590953-A1 TETRAZOLE COMPOUNDS AS CALCIUM CHANNEL BLOCKERS Convergence Pharmaceuticals Limited (GB) 2013-05-15 EP disclosed
WO-2012004604-A1 TETRAZOLE COMPOUNDS AS CALCIUM CHANNEL BLOCKERS Convergence Pharmaceuticals Limited (GB) 2012-01-12 WO disclosed