SCHEMBL12605459

SCHEMBL12605459

CS(=O)(=O)NCCCc1c[nH]c2nccnc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.43
MAPK1 P28482 1/20 0.38
CDC7 O00311 1/20 0.35
DAPK3 O43293 1/20 0.35
ROCK2 O75116 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35
PAK4 O96013 1/20 0.35
PIM1 P11309 1/20 0.35
PRKACA P17612 1/20 0.35
CDK2 P24941 1/20 0.35
FLT3 P36888 1/20 0.35
CSNK1A1 P48729 1/20 0.35
CDK8 P49336 1/20 0.35
CLK2 P49760 1/20 0.35
GSK3B P49841 1/20 0.35
CDK7 P50613 1/20 0.35
CDK9 P50750 1/20 0.35
PRKX P51817 1/20 0.35
JAK3 P52333 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12605488 0.78 ALOX12 (0.33) CDK2ALDH1A1MTNR1AALOX12HTR1A
SCHEMBL12605483 0.78 ALDH1A1 (0.43) ALDH1A1NPY5RMAPT
SCHEMBL12605462 0.78 MTNR1A (0.54) ALDH1A1MTNR1ANQO2KDM4EMAPT
SCHEMBL12605492 0.78 CYP2D6 (0.51) POLBALDH1A1NPY5RKDM4EHTT
SCHEMBL12605447 0.74 MAPK1 (0.44) MAPK1CDK2MTNR1AGPR84SLC6A4
SCHEMBL12605470 0.74 MAPK1 (0.44) MAPK1CDK2GPR84HTR1ASLC6A4
SCHEMBL12605481 0.74 MTNR1A (0.47) MTNR1AGPR84
SCHEMBL12244242 0.73 MAPK1 (0.50) MAPK1CDC7MAP4K4PAK4CDK2
SCHEMBL12605484 0.73 MTNR1A (0.38) MAPK1ALDH1A1MTNR1AKDM4EHSD17B10
SCHEMBL12605482 0.73 SPR (0.46) MTNR1AMAPTHSD17B10HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7943616-B2 Protein kinase inhibitors; astham; psoriasis; antiinflammatory agents; inflammatory bowel disorders AVENTIS PHARMACEUTICALS INC. (US) 2011-05-17 US disclosed
US-7227020-B2 Azaindoles AVENTIS PHARMA LIMITED (GB) 2007-06-05 US disclosed